SCHEMBL8666291

SCHEMBL8666291

O=C(O)N1CCN(CCc2ccc([N+](=O)[O-])cc2)CC1

nearest known ligand 0.77

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
KCNJ1 P48048 14/20 0.77
KCNH2 Q12809 13/20 0.77
HRH3 Q9Y5N1 1/20 0.68
SIGMAR1 Q99720 2/20 0.67
HTR2A P28223 1/20 0.57
MAOA P21397 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2731306 0.88 KCNJ1 (1.00) KCNJ1KCNH2HRH3SIGMAR1MAOA
SCHEMBL27555522 0.87 KCNJ1 (0.75) KCNJ1KCNH2HRH3SIGMAR1MAOA
SCHEMBL8509511 0.86 KCNJ1 (0.77) KCNJ1KCNH2HRH3SIGMAR1HTR2A
SCHEMBL8715859 0.86 KCNJ1 (0.77) KCNJ1KCNH2HRH3SIGMAR1HTR2A
SCHEMBL6416345 0.85 KDM4E (0.71) KCNJ1
SCHEMBL4717096 0.84 SIGMAR1 (0.71) KCNJ1KCNH2SIGMAR1HTR2A
SCHEMBL286800 0.84 KCNJ1 (0.84) KCNJ1KCNH2HRH3SIGMAR1MAOA
SCHEMBL17444701 0.83 KCNH2 (0.73) KCNJ1KCNH2HRH3SIGMAR1HTR2A
SCHEMBL3526680 0.82 KCNJ1 (0.87) KCNJ1KCNH2HRH3SIGMAR1MAOA
SCHEMBL5653299 0.82 HRH3 (0.93) KCNJ1KCNH2HRH3SIGMAR1MAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0880512-A1 NOVEL AROMATIC PIPERAZINES DERIVED FROM SUBSTITUTED CYCLOAZANES, METHOD FOR PREPARING SAME, PHARMACEUTICAL COMPOSITIONS, AND USE THEREOF AS DRUGS PIERRE FABRE MEDICAMENT (FR) 1998-12-02 EP disclosed
WO-1997028141-A1 NOVEL AROMATIC PIPERAZINES DERIVED FROM SUBSTITUTED CYCLOAZANES, METHOD FOR PREPARING SAME, PHARMACEUTICAL COMPOSITIONS, AND USE THEREOF AS DRUGS PIERRE FABRE MEDICAMENT (FR) 1997-08-07 WO disclosed