SCHEMBL8670044

SCHEMBL8670044

CC(C)c1cc(/C=C2/CCON(C)C2=O)cc(C(C)C)c1O

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 3/20 0.59
CYP3A4 P08684 3/20 0.59
CYP2B6 P20813 2/20 0.59
PTGS2 P35354 3/20 0.39
PTGS1 P23219 2/20 0.39
ALOX5 P09917 1/20 0.39
EGFR P00533 3/20 0.38
ERBB2 P04626 2/20 0.38
PDGFRB P09619 2/20 0.38
IGF1R P08069 1/20 0.38
NOX4 Q9NPH5 1/20 0.38
GLRA1 P23415 1/20 0.36
CYP2C9 P11712 3/20 0.36
MAPT P10636 2/20 0.35
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
KDM4E B2RXH2 1/20 0.34
MEN1 O00255 1/20 0.34
LMNA P02545 1/20 0.34
POLB P06746 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8670047 1.00 CYP1A2 (0.59) CYP1A2CYP3A4CYP2B6PTGS2PTGS1
SCHEMBL2682345 0.80 CYP1A2 (0.58) CYP1A2CYP3A4CYP2B6PTGS2PTGS1
SCHEMBL2681961 0.79 PTGS1 (0.64) CYP1A2PTGS2PTGS1ALOX5EGFR
SCHEMBL2681962 0.79 PTGS1 (0.64) CYP1A2PTGS2PTGS1ALOX5EGFR
SCHEMBL8291651 0.79 PTGS1 (0.64) CYP1A2PTGS2PTGS1ALOX5EGFR
SCHEMBL11129914 0.78 CYP1A2 (0.66) CYP1A2CYP3A4CYP2B6PTGS2PTGS1
SCHEMBL13178556 0.75 CYP1A2 (0.46) CYP1A2CYP3A4CYP2B6PTGS2PTGS1
SCHEMBL8779681 0.74 CYP1A2 (0.59) CYP1A2CYP3A4CYP2B6PTGS2PTGS1
SCHEMBL8779682 0.74 CYP1A2 (0.59) CYP1A2CYP3A4CYP2B6PTGS2PTGS1
SCHEMBL8779692 0.71 CYP1A2 (0.56) CYP1A2CYP3A4CYP2B6PTGS2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0830133-A1 THERAPEUTIC COMPOSITION FOR ARTHRITIS Takeda Chemical Industries, Ltd. (JP) 1998-03-25 EP disclosed
WO-1996033717-A1 THERAPEUTIC COMPOSITION FOR ARTHRITIS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1996-10-31 WO disclosed