SCHEMBL8670858

SCHEMBL8670858

CS(=O)(=O)NC1CCN(c2cc(C(F)(F)F)ccn2)C1=O

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP17A1 P05093 1/20 0.47
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41
MAPT P10636 1/20 0.41
CA12 O43570 1/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CA9 Q16790 1/20 0.41
ADRB1 P08588 1/20 0.41
SMO Q99835 1/20 0.41
CXCR3 P49682 1/20 0.41
NR1H2 P55055 1/20 0.40
NR1H3 Q13133 1/20 0.40
MAP3K12 Q12852 3/20 0.39
CCR2 P41597 2/20 0.39
CCR5 P51681 1/20 0.39
FFAR4 Q5NUL3 1/20 0.39
GAA P10253 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
CYP11B1 P15538 2/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8787300 0.86 CYP17A1 (0.51) CYP17A1KDM4EALDH1A1MAPTCA12
SCHEMBL13063399 0.79 CYP17A1 (0.51) CYP17A1KDM4EALDH1A1MAPTADRB1
SCHEMBL13018940 0.77 CYP17A1 (0.49) CYP17A1KDM4EALDH1A1MAPTADRB1
SCHEMBL8789168 0.77 CYP17A1 (0.51) CYP17A1KDM4EALDH1A1MAPTADRB1
SCHEMBL9265494 0.77 CYP17A1 (0.54) CYP17A1KDM4EALDH1A1MAPTADRB1
SCHEMBL8789598 0.76 CNR1 (0.43) CYP17A1KDM4EALDH1A1MAPTADRB1
SCHEMBL8658729 0.76 CYP17A1 (0.43) CYP17A1KDM4EALDH1A1MAPTADRB1
SCHEMBL13063691 0.74 CYP17A1 (0.46) CYP17A1KDM4EMAPTADRB1CXCR3
SCHEMBL8661026 0.72 CNR1 (0.45) CYP17A1KDM4EALDH1A1MAPTADRB1
SCHEMBL13063400 0.69 CYP17A1 (0.56) CYP17A1KDM4EALDH1A1MAPTADRB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0828710-A1 PROCESS FOR THE PREPARATION OF (THIO-)CARBONIC/CARBAMIC ACID 2-PYRROLIDONYL-3-ESTERS, THIO ESTERS AND AMIDES ZENECA LIMITED (GB) 1998-03-18 EP disclosed
WO-1996037466-A1 PROCESS FOR THE PREPARATION OF (THIO-)CARBONIC/CARBAMIC ACID 2-PYRROLIDONYL-3-ESTERS, THIO ESTERS AND AMIDES ZENECA LIMITED (GB) 1996-11-28 WO disclosed