SCHEMBL8670880

SCHEMBL8670880

CC(=O)Sc1ccc2ccccc2c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EPHX1 P07099 1/20 0.51
ANPEP P15144 1/20 0.47
CES2 O00748 1/20 0.47
CES1 P23141 1/20 0.47
KDM4E B2RXH2 3/20 0.44
SMN1; SMN2 Q16637 3/20 0.44
HPGD P15428 2/20 0.44
ALDH1A1 P00352 3/20 0.43
CYP1A2 P05177 2/20 0.43
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
CYP2C19 P33261 1/20 0.43
HIF1A Q16665 1/20 0.43
SIRT2 Q8IXJ6 1/20 0.41
SIRT1 Q96EB6 1/20 0.41
SIRT3 Q9NTG7 1/20 0.41
TDP1 Q9NUW8 2/20 0.41
CYP2A6 P11509 1/20 0.41
CA12 O43570 1/20 0.41
CA1 P00915 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29282031 0.87 AKR1C3 (0.38) EPHX1ANPEPKDM4EHPGDALDH1A1
SCHEMBL1479596 0.81 ANPEP (0.49) EPHX1ANPEPCES2CES1KDM4E
SCHEMBL29267422 0.80 EPHX1 (0.45) EPHX1ANPEPCES2CES1KDM4E
SCHEMBL1403189 0.79 ANPEP (0.47) EPHX1ANPEPCES2CES1KDM4E
SCHEMBL9666253 0.79 EPHX1 (0.56) EPHX1ANPEPCES2CES1KDM4E
SCHEMBL11332669 0.79 ALDH1A1 (0.50) EPHX1ANPEPCES2CES1KDM4E
SCHEMBL11764204 0.79 ANPEP (0.47) EPHX1ANPEPCES2CES1KDM4E
SCHEMBL28340440 0.78 ANPEP (0.46) EPHX1ANPEPCES2CES1KDM4E
SCHEMBL22958258 0.78 EPHX1 (0.42) EPHX1ANPEPCES2CES1KDM4E
SCHEMBL14341653 0.77 HPGD (0.46) HPGDALDH1A1MEN1KMT2ACA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109796383-B 1-thiophenyl-N-acetyl-2-naphthylamine and its derivative and synthesis method 湘潭大学 2020-09-18 CN claimed
CN-109796383-B 1-thiophenyl-N-acetyl-2-naphthylamine and its derivative and synthesis method 湘潭大学 2020-09-18 CN disclosed
CN-110536884-A synthesis of MCL-1 inhibitors ASTRAZENECA AB 2019-12-03 CN disclosed
US-5710211-A REACTION OF POLYMER WITH COMPOUND HAVING A THIOL OR THIOESTER AND HYDROLYSIS TO FORM VINYL ALCOHOL KURARAY CO., LTD. (JP) 1998-01-20 US disclosed