SCHEMBL8673448

SCHEMBL8673448

COc1cc(C(=O)N(C)c2ccc(C)cc2OCCCCC(=C=O)N2CCC(N(C)C)CC2)ccc1NC(=O)c1cccc(OCCCNC(=O)OC(C)(C)C)c1

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 1/20 0.36
FYN P06241 1/20 0.36
SRC P12931 1/20 0.36
PTK6 Q13882 1/20 0.36
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
PRKAA2 P54646 1/20 0.34
PTK2 Q05397 1/20 0.34
AVPR2 P30518 1/20 0.33
AVPR1A P37288 1/20 0.33
AVPR1B P47901 1/20 0.33
ADRA1D P25100 4/20 0.33
ADRA1A P35348 4/20 0.33
ADRA1B P35368 4/20 0.33
DRD2 P14416 2/20 0.33
DRD4 P21917 2/20 0.33
DRD3 P35462 2/20 0.33
POLB P06746 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7339013 0.93 AVPR2 (0.38) ABL1FYNSRCPTK6MEN1
SCHEMBL7339138 0.85 AVPR2 (0.43) ABL1FYNSRCPTK6KMT2A
SCHEMBL7340438 0.82 ABL1 (0.38) ABL1FYNSRCPTK6KMT2A
Hydrochloric Acid SCHEMBL7336979 0.82 AVPR2 (0.40) MEN1KMT2APTK2AVPR2AVPR1A
SCHEMBL7337083 0.80 AVPR2 (0.43) ABL1FYNSRCPTK6AVPR2
SCHEMBL7338676 0.80 AVPR2 (0.40) AVPR2AVPR1AAVPR1BADRA1DADRA1A
SCHEMBL7342434 0.80 AVPR2 (0.42) KMT2AAVPR2AVPR1AAVPR1B
Hydrochloric Acid SCHEMBL7780856 0.80 AVPR2 (0.39) AVPR2AVPR1AAVPR1BADRA1DADRA1A
SCHEMBL7338448 0.79 AVPR2 (0.37) MEN1KMT2AAVPR2AVPR1AAVPR1B
SCHEMBL7340542 0.79 AVPR2 (0.37) KMT2AAVPR2AVPR1AAVPR1BADRA1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0832061-A1 BENZAMIDE DERIVATIVES AND THEIR USE AS VASOPRESSIN ANTAGONISTS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 1998-04-01 EP disclosed