SCHEMBL8675878

SCHEMBL8675878

CC(C)(C)OC(=O)Nc1cc(-c2ccc(C(Br)Br)cc2)ccn1

nearest known ligand 0.46

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
AAK1 Q2M2I8 14/20 0.46
CYP3A4 P08684 3/20 0.45
GSK3B P49841 1/20 0.45
DYRK1A Q13627 1/20 0.45
IRAK4 Q9NWZ3 1/20 0.44
CYP17A1 P05093 2/20 0.43
MAP4K4 O95819 1/20 0.42
PIK3C3 Q8NEB9 1/20 0.42
ROCK2 O75116 1/20 0.42
NR2C2 P49116 1/20 0.42
MAP2K1 Q02750 1/20 0.42
HIPK4 Q8NE63 1/20 0.42
CLK4 Q9HAZ1 1/20 0.42
BMP2K Q9NSY1 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8670718 0.85 FDPS (0.50) AAK1CYP3A4GSK3BDYRK1AIRAK4
SCHEMBL5251219 0.83 EGFR (0.57) AAK1GSK3BDYRK1AIRAK4CYP17A1
SCHEMBL9232528 0.83 CYP17A1 (0.50) AAK1CYP3A4GSK3BDYRK1AIRAK4
SCHEMBL12127932 0.82 FDPS (0.54) AAK1GSK3BDYRK1APIK3C3
SCHEMBL5544966 0.82 CYP17A1 (0.47) AAK1CYP3A4GSK3BDYRK1AIRAK4
SCHEMBL5251601 0.81 GSK3B (0.46) AAK1CYP3A4GSK3BDYRK1AIRAK4
SCHEMBL5548970 0.81 ATR (0.48) AAK1CYP3A4GSK3BDYRK1AIRAK4
SCHEMBL29992322 0.80 AAK1 (0.48) AAK1CYP3A4GSK3BDYRK1AIRAK4
SCHEMBL17643492 0.80 AAK1 (0.48) AAK1CYP3A4GSK3BDYRK1AIRAK4
SCHEMBL27955914 0.80 ATR (0.42) AAK1GSK3BDYRK1AIRAK4CYP17A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5854245-A Fibrinogen receptor antagonists MERCK & CO., INC. (US) 1998-12-29 US disclosed