Spermine

Spermine

SCHEMBL867751

NCCCNCCCCNCCCN.O=P(O)(O)O.O=P(O)(O)O

nearest known ligand 0.68

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ADRA1AADRA1BADRA1DADRB1ADRB2ADRB3CYP11B1DPP4FGFR1FGFR2FGFR3FGFR4HRH1JAK1JAK2JAK3KCNA1KCNA10KCNA2KCNA3KCNA4KCNA5KCNA6KCNA7KCNB1KCNB2KCNC1KCNC2KCNC3KCNC4KCND1KCND2KCND3KCNF1KCNG1KCNG2KCNG3KCNG4KCNH1KCNH2KCNH3KCNH4KCNH5KCNH6KCNH7KCNH8KCNQ1KCNQ2KCNQ3KCNQ4KCNQ5KCNS1KCNS2KCNS3KCNV1KCNV2KDRKITNAOPRD1OPRK1OPRM1PPDGFRBPIK3CDSCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASMOTYK2polrplArplBrplCrplDrplErplFrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmFrpmGrpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of Spermine. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 3/20 0.68
CA2 P00918 3/20 0.68
CA4 P22748 3/20 0.68
CA6 P23280 3/20 0.68
CA5A P35218 3/20 0.68
CA7 P43166 3/20 0.68
CA9 Q16790 3/20 0.68
CA14 Q9ULX7 3/20 0.68
CA5B Q9Y2D0 3/20 0.68
F13A1 P00488 2/20 0.68
CYP1A2 P05177 2/20 0.68
ALOX15 P16050 2/20 0.68
THPO P40225 2/20 0.68
CASP2 P42575 2/20 0.68
MEN1 O00255 1/20 0.68
CYP2C19 P33261 1/20 0.68
RECQL P46063 1/20 0.68
KMT2A Q03164 1/20 0.68
HSD17B10 Q99714 1/20 0.68
CA3 P07451 2/20 0.65

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Spermine SCHEMBL2058654 1.00 CA12 (0.68) CA12CA2CA4CA6CA5A
Spermidine SCHEMBL867617 0.97 CA12 (0.70) CA12CA2CA4CA6CA5A
Spermine SCHEMBL364155 0.97 CA12 (0.65) CA12CA2CA4CA6CA5A
Spermidine SCHEMBL343200 0.95 CA12 (0.67) CA12CA2CA4CA6CA5A
Spermidine SCHEMBL28472688 0.95 CA12 (0.67) CA12CA2CA4CA6CA5A
Phosphoric Acid SCHEMBL15512587 0.92 CA12 (0.62) CA12CA2CA4CA6CA5A
Phosphoric Acid SCHEMBL5552800 0.86 CA12 (0.54) CA12CA2CA4CA6CA5A
Phosphoric Acid SCHEMBL5548350 0.86 CA12 (0.54) CA12CA2CA4CA6CA5A
Spermine SCHEMBL867750 0.86 CA12 (0.56) CA12CA2CA4CA6CA5A
Wr-1065 SCHEMBL1821959 0.86 ESR1 (0.74) CA12CA2CA4CA6CA5A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 20 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3122759-B1 CHEMICAL METHODS FOR PRODUCING TAGGED NUCLEOTIDES UNIV COLUMBIA (US) 2022-06-01 EP disclosed
EP-2289863-B1 Environmental barrier coatings for high temperature ceramic components GEN ELECTRIC (US) 2020-11-18 EP disclosed
EP-2287131-B1 Slurry-derived environmental barrier coatings GEN ELECTRIC (US) 2020-09-02 EP disclosed
EP-2287132-B1 Methods for making environmental barrier coatings using sintering aids GEN ELECTRIC (US) 2019-08-28 EP disclosed
EP-2287129-B1 Methods of improving surface roughness of an environmental barrier coating GEN ELECTRIC (US) 2016-09-07 EP disclosed
US-9212100-B2 Environmental barrier coatings for high temperature ceramic components GENERAL ELECTRIC COMPANY (US) 2015-12-15 US disclosed
US-9073793-B2 Slurry compositions for making environmental barrier coatings and environmental barrier coatings comprising the same GENERAL ELECTRIC COMPANY (US) 2015-07-07 US disclosed
US-9056802-B2 Methods for making environmental barrier coatings using sintering aids GENERAL ELECTRIC COMPANY (US) 2015-06-16 US disclosed
US-8986779-B2 Methods of improving surface roughness of an environmental barrier coating and components comprising environmental barrier coatings having improved surface roughness GENERAL ELECTRIC COMPANY (US) 2015-03-24 US disclosed
US-20120076943-A1 METHODS FOR MAKING ENVIRONMENTAL BARRIER COATINGS USING SINTERING AIDS DEPARTMENT OF THE NAVY 2012-03-29 US disclosed
US-20120077004-A1 ENVIRONMENTAL BARRIER COATINGS FOR HIGH TEMPERATURE CERAMIC COMPONENTS DEPARTMENT OF THE NAVY 2012-03-29 US disclosed
US-20110229632-A1 METHODS OF IMPROVING SURFACE ROUGHNESS OF AN ENVIRONMENTAL BARRIER COATING AND COMPONENTS COMPRISING ENVIRONMENTAL BARRIER COATINGS HAVING IMRPOVED SURFACE ROUGHNESS DEPARTMENT OF THE NAVY 2011-09-22 US disclosed
EP-2289863-A2 Environmental barrier coatings for high temperature ceramic components General Electric Company (US) 2011-03-02 EP disclosed
EP-2287130-A2 Methods of making environmental barrier coatings for high temperature ceramic components using sintering aids General Electric Company (US) 2011-02-23 EP disclosed
EP-2287132-A2 Methods for making environmental barrier coatings using sintering aids General Electric Company (US) 2011-02-23 EP disclosed
EP-2287129-A2 Methods of improving surface roughness of an environmental barrier coating General Electric Company (US) 2011-02-23 EP disclosed
EP-2287131-A2 Slurry compositions for making environmental barrier coatings and environmental barrier coatings comprising the same General Electric Company (US) 2011-02-23 EP disclosed
US-20110027467-A1 METHODS OF MAKING ENVIRONMENTAL BARRIER COATINGS FOR HIGH TEMPERATURE CERAMIC COMPONENTS USING SINTERING AIDS GENERAL ELECTRIC COMPANY 2011-02-03 US disclosed
US-20110027556-A1 SLURRY COMPOSITIONS FOR MAKING ENVIRONMENTAL BARRIER COATINGS AND ENVIRONMENTAL BARRIER COATINGS COMPRISING THE SAME DEPARTMENT OF THE NAVY 2011-02-03 US disclosed
US-4957757-A Method of extending shelf life and enhancing keeping quality of fruits CORNELL RESEARCH FOUNDATION, INC. (US) 1990-09-18 US disclosed