SCHEMBL8677779

SCHEMBL8677779

Cc1ccc(N=C=O)cc1[N+](=O)[O-].O=C=Nc1ccc(Cl)cc1[N+](=O)[O-]

nearest known ligand 0.49

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.49
TRPA1 O75762 1/20 0.49
MPI P34949 1/20 0.44
CCR2 P41597 3/20 0.41
VCAM1 P19320 1/20 0.40
TSHR P16473 3/20 0.39
ALDH1A1 P00352 1/20 0.39
RECQL P46063 1/20 0.39
HSP90AA1 P07900 1/20 0.38
TDP1 Q9NUW8 3/20 0.38
MAPK1 P28482 2/20 0.38
LMNA P02545 1/20 0.37
MAPT P10636 3/20 0.36
GAA P10253 1/20 0.36
PPIA P62937 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3842281 0.85 VCAM1 (0.51) VCAM1TSHRALDH1A1MAPK1LMNA
SCHEMBL61198 0.85 CYP3A4 (0.56) CYP3A4TRPA1MPITSHRALDH1A1
SCHEMBL29389795 0.84 CYP3A4 (0.49) CYP3A4TRPA1TSHRALDH1A1TDP1
SCHEMBL124224 0.84 CYP3A4 (0.49) CYP3A4TRPA1TSHRALDH1A1TDP1
SCHEMBL10718338 0.78 CYP3A4 (0.47) CYP3A4TRPA1TSHRALDH1A1TDP1
SCHEMBL8735930 0.78 VCAM1 (0.53) VCAM1TSHRALDH1A1MAPK1LMNA
SCHEMBL30976988 0.78 TSHR (0.60) CYP3A4CCR2VCAM1TSHRALDH1A1
SCHEMBL400340 0.78 TSHR (0.60) CYP3A4CCR2VCAM1TSHRALDH1A1
Methyl Alcohol SCHEMBL28263562 0.74 TSHR (0.56) CYP3A4CCR2VCAM1TSHRALDH1A1
SCHEMBL3839311 0.73 CYP3A4 (0.56) CYP3A4TRPA1MPITSHRALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0880558-A1 COMBINATORIAL PROCESS FOR PREPARING SUBSTITUTED INDANE LIBRARIES ELI LILLY AND COMPANY (US) 1998-12-02 EP disclosed
WO-1998008813-A1 COMBINATORIAL PROCESS FOR PREPARING SUBSTITUTED PYRROLIDINE LIBRARIES ELI LILLY AND COMPANY (US) 1998-03-05 WO disclosed
WO-1997026300-A1 COMBINATORIAL PROCESS FOR PREPARING SUBSTITUTED INDANE LIBRARIES ELI LILLY AND COMPANY (US) 1997-07-24 WO disclosed