SCHEMBL8680461

SCHEMBL8680461

C=CCOC(=O)c1nc(C#N)c[nH]1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.41
ALDH1A1 P00352 5/20 0.36
HSD17B10 Q99714 4/20 0.36
TSHR P16473 2/20 0.36
SNCA P37840 1/20 0.36
KDM4E B2RXH2 7/20 0.35
MAPT P10636 6/20 0.35
MEN1 O00255 4/20 0.35
KMT2A Q03164 4/20 0.35
LMNA P02545 2/20 0.35
TP53 P04637 2/20 0.35
ALOX15 P16050 1/20 0.35
CASP1 P29466 1/20 0.35
GAA P10253 1/20 0.34
CYP1A2 P05177 2/20 0.34
CYP2D6 P10635 2/20 0.34
CYP2C9 P11712 2/20 0.34
CYP2C19 P33261 2/20 0.34
NPSR1 Q6W5P4 2/20 0.33
HTT P42858 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8680459 0.70 MYC (0.35)
SCHEMBL16118350 0.70 AHR (0.33) ALDH1A1HSD17B10KDM4EMAPTHTT
SCHEMBL19868327 0.69 CREBBP (0.35) TSHRHTTHPGDSMN1; SMN2
SCHEMBL3558245 0.69 KMT2A (0.50) CYP3A4ALDH1A1HSD17B10TSHRSNCA
SCHEMBL7592184 0.69 CYP3A4 (0.41) CYP3A4ALDH1A1HSD17B10TSHRSNCA
SCHEMBL3034729 0.68 CYP3A4 (0.46) CYP3A4ALDH1A1HSD17B10TSHRSNCA
SCHEMBL19264828 0.66
SCHEMBL3601302 0.66 SNCA (0.44) CYP3A4ALDH1A1HSD17B10TSHRSNCA
SCHEMBL6230747 0.65 SNCA (0.54) CYP3A4ALDH1A1HSD17B10TSHRSNCA
SCHEMBL5868399 0.64 CYP3A4 (0.45) CYP3A4ALDH1A1HSD17B10TSHRSNCA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5750692-A Synthesis of 3-deazapurines ISIS PHARMACEUTICALS, INC. (US) 1998-05-12 US claimed