SCHEMBL8680459

SCHEMBL8680459

N#Cc1c[nH]c(C(N)=O)n1

nearest known ligand 0.35

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
MYC P01106 1/20 0.35
CHUK O15111 2/20 0.34
AHR P35869 1/20 0.33
PARP15 Q460N3 1/20 0.33
PARP10 Q53GL7 1/20 0.33
PARP2 Q9UGN5 1/20 0.33
PARP1 P09874 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1863248 0.82 PIN1 (0.39) AHR
SCHEMBL16118350 0.81 AHR (0.33) AHR
SCHEMBL19264828 0.81
SCHEMBL19868327 0.77 CREBBP (0.35) AHR
SCHEMBL3821371 0.73 LMNA (0.41)
SCHEMBL161337 0.71
SCHEMBL8561 0.71
SCHEMBL161336 0.71
SCHEMBL15436573 0.71 POLB (0.45)
SCHEMBL8680461 0.70 CYP3A4 (0.41)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5750692-A Synthesis of 3-deazapurines ISIS PHARMACEUTICALS, INC. (US) 1998-05-12 US claimed
EP-3208269-A1 INHIBITORS OF C-FMS KINASE Janssen Pharmaceutica N.V. (BE) 2017-08-23 EP disclosed
EP-1807077-B1 INHIBITORS OF C-FMS KINASE JANSSEN PHARMACEUTICA NV (BE) 2016-11-23 EP disclosed
EP-2687516-A1 Inhibitors of C-FMS Kinase Janssen Pharmaceutica N.V. (BE) 2014-01-22 EP disclosed