SCHEMBL8683285

SCHEMBL8683285

Cc1cc[n+]([O-])c(C)c1O

nearest known ligand 0.40

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.40
KDM4E B2RXH2 2/20 0.37
MAPT P10636 1/20 0.37
TRPA1 O75762 1/20 0.36
CCR5 P51681 1/20 0.35
GABRA1 P14867 1/20 0.31
GABRB2 P47870 1/20 0.31
HPGD P15428 1/20 0.30
HSD17B10 Q99714 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL316864 0.77 DPP4 (0.30)
SCHEMBL667046 0.75 CCR5 (0.33) CCR5
SCHEMBL2722030 0.71 CCR5 (0.32) CCR5
SCHEMBL11421873 0.71 CCR5 (0.32) ALDH1A1CCR5
SCHEMBL2085322 0.71 CCR5 (0.44) ALDH1A1CCR5
SCHEMBL10073293 0.68 CCR5 (0.31) CCR5
SCHEMBL13145619 0.68 CCR5 (0.31) CCR5
SCHEMBL13542937 0.67 CCR5 (0.42) CCR5
SCHEMBL14272580 0.67 CCR5 (0.42) ALDH1A1KDM4ECCR5
SCHEMBL3319954 0.67

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5721259-A Method of using 2-formylpyridine thiosemicarbazone compounds YALE UNIVERSITY (US) 1998-02-24 US disclosed
EP-0570294-B1 2-Formylpyridine thiosemicarbazone derivatives, their preparation and their use as antitumor agents UNIV YALE (US) 1997-07-30 EP disclosed
US-5281715-A 2-formylpyridine thiosemicarbazone compounds YALE UNIVERSITY (US) 1994-01-25 US disclosed
EP-0570294-A1 2-Formylpyridine thiosemicarbazone derivatives, their preparation and their use as antitumor agents YALE UNIVERSITY (US) 1993-11-18 EP disclosed