SCHEMBL8683501

SCHEMBL8683501

CC(=O)Nc1cnc(C=NNC(N)=S)cc1C

nearest known ligand 0.49

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
RRM2 P31350 9/20 0.48
MEN1 O00255 3/20 0.41
KMT2A Q03164 3/20 0.41
ALDH1A1 P00352 3/20 0.41
L3MBTL1 Q9Y468 2/20 0.41
MAPT P10636 2/20 0.41
USP2 O75604 1/20 0.41
GAA P10253 1/20 0.41
NCOA1 Q15788 2/20 0.40
NCOA3 Q9Y6Q9 2/20 0.40
G6PD P11413 1/20 0.40
KDM4E B2RXH2 3/20 0.39
NPC1 O15118 1/20 0.39
OPRK1 P41145 1/20 0.39
HTT P42858 1/20 0.39
RAB9A P51151 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
LMNA P02545 1/20 0.39
HPGD P15428 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31753303 0.84 RRM2 (0.52) RRM2MEN1KMT2AALDH1A1L3MBTL1
SCHEMBL4390542 0.84 RRM2 (0.52) RRM2MEN1KMT2AALDH1A1L3MBTL1
SCHEMBL8683429 0.81 RRM2 (0.47) RRM2MEN1KMT2AALDH1A1L3MBTL1
SCHEMBL6264236 0.79 RRM2 (0.55) RRM2MEN1KMT2AALDH1A1L3MBTL1
SCHEMBL4380310 0.79 RRM2 (0.55) RRM2MEN1KMT2AALDH1A1L3MBTL1
SCHEMBL6264240 0.79 RRM2 (0.55) RRM2MEN1KMT2AALDH1A1L3MBTL1
SCHEMBL6261112 0.77 RRM2 (0.71) RRM2MEN1KMT2AALDH1A1NCOA1
SCHEMBL6261110 0.77 RRM2 (0.71) RRM2MEN1KMT2AALDH1A1NCOA1
SCHEMBL8689525 0.76 LMNA (0.45) RRM2MEN1KMT2AALDH1A1L3MBTL1
SCHEMBL8682966 0.75 RRM2 (0.44) RRM2ALDH1A1MAPTGAANCOA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5721259-A Method of using 2-formylpyridine thiosemicarbazone compounds YALE UNIVERSITY (US) 1998-02-24 US disclosed
EP-0570294-B1 2-Formylpyridine thiosemicarbazone derivatives, their preparation and their use as antitumor agents UNIV YALE (US) 1997-07-30 EP disclosed
US-5281715-A 2-formylpyridine thiosemicarbazone compounds YALE UNIVERSITY (US) 1994-01-25 US disclosed
EP-0570294-A1 2-Formylpyridine thiosemicarbazone derivatives, their preparation and their use as antitumor agents YALE UNIVERSITY (US) 1993-11-18 EP disclosed