SCHEMBL8684157

SCHEMBL8684157

CC(C)(C)CN1C(=O)[C@@H](CC(=O)O)S[C@H](c2cccc3ccccc23)c2cc(Br)ccc21

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.39
MAPT P10636 3/20 0.37
TP53 P04637 2/20 0.37
TSHR P16473 2/20 0.35
KDM4E B2RXH2 1/20 0.35
HTT P42858 1/20 0.35
CDC25A P30304 1/20 0.34
FDFT1 P37268 1/20 0.33
XIAP P98170 1/20 0.33
POLB P06746 1/20 0.33
KMT2A Q03164 2/20 0.32
MEN1 O00255 1/20 0.32
TDP2 O95551 1/20 0.32
CFTR P13569 1/20 0.32
CASP6 P55212 1/20 0.32
HKDC1 Q2TB90 1/20 0.32
GOPC Q9HD26 1/20 0.32
GAA P10253 1/20 0.32
BACE1 P56817 1/20 0.32
GSK3B P49841 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8684153 1.00 ALDH1A1 (0.39) ALDH1A1MAPTTP53TSHRKDM4E
SCHEMBL8684150 1.00 ALDH1A1 (0.39) ALDH1A1MAPTTP53TSHRKDM4E
SCHEMBL8684377 0.90 GSK3B (0.36) ALDH1A1MAPTTP53KDM4EHTT
SCHEMBL8684371 0.90 GSK3B (0.36) ALDH1A1MAPTTP53KDM4EHTT
SCHEMBL8684367 0.90 GSK3B (0.36) ALDH1A1MAPTTP53KDM4EHTT
SCHEMBL8636201 0.89 FDFT1 (0.43) ALDH1A1MAPTHTTFDFT1
SCHEMBL8636199 0.89 FDFT1 (0.43) ALDH1A1MAPTHTTFDFT1
SCHEMBL8636205 0.89 FDFT1 (0.43) ALDH1A1MAPTHTTFDFT1
SCHEMBL8686109 0.88 ALDH1A1 (0.34) ALDH1A1MAPTTSHRKDM4EHTT
SCHEMBL8686114 0.88 ALDH1A1 (0.34) ALDH1A1MAPTTSHRKDM4EHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5770594-A ANTICHOLESTEROL AGENTS, INHIBITORS OF CHOLESTEROL SYNTHESIS PFIZER INC. (US) 1998-06-23 US disclosed
WO-1996020184-A1 NAPHTHYL-BENZOXAZEPINES OR -BENZOTHIAZEPINES AS SQUALENE SYNTHETASE INHIBITORS PFIZER INC. (US) 1996-07-04 WO disclosed