SCHEMBL8685653

SCHEMBL8685653

NC(=S)NN=Cc1ccc([N+](=O)[O-])cn1

nearest known ligand 0.64

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.64
MAOB P27338 1/20 0.64
SLC2A1 P11166 1/20 0.61
RRM2 P31350 6/20 0.58
HTT P42858 1/20 0.57
MEN1 O00255 4/20 0.53
KMT2A Q03164 4/20 0.53
ALDH1A1 P00352 3/20 0.53
GAA P10253 1/20 0.51
CTDSP1 Q9GZU7 1/20 0.49
KDM4E B2RXH2 1/20 0.48
OPRK1 P41145 1/20 0.48
ADRA2A P08913 1/20 0.47
ADRA2B P18089 1/20 0.47
ADRA2C P18825 1/20 0.47
LMNA P02545 1/20 0.46
HPGD P15428 1/20 0.46
ALOX12 P18054 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29420113 0.77 RRM2 (0.67) RRM2GAAKDM4E
SCHEMBL783293 0.77 RRM2 (0.67) RRM2GAAKDM4E
SCHEMBL783292 0.77 RRM2 (0.67) RRM2GAAKDM4E
SCHEMBL31753656 0.77 RRM2 (0.67) RRM2KDM4E
SCHEMBL4382591 0.77 RRM2 (0.67) RRM2KDM4E
SCHEMBL30094126 0.77 RRM2 (0.67) RRM2GAAKDM4E
SCHEMBL7749775 0.77 RRM2 (0.67) RRM2KDM4E
SCHEMBL25042631 0.76 SLC2A1 (1.00) MAPTSLC2A1MEN1KMT2AALDH1A1
SCHEMBL30275111 0.76 SLC2A1 (1.00) MAPTSLC2A1MEN1KMT2AALDH1A1
SCHEMBL30275251 0.76 SLC2A1 (1.00) MAPTSLC2A1MEN1KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5721259-A Method of using 2-formylpyridine thiosemicarbazone compounds YALE UNIVERSITY (US) 1998-02-24 US disclosed
EP-0570294-B1 2-Formylpyridine thiosemicarbazone derivatives, their preparation and their use as antitumor agents UNIV YALE (US) 1997-07-30 EP disclosed
US-5281715-A 2-formylpyridine thiosemicarbazone compounds YALE UNIVERSITY (US) 1994-01-25 US disclosed
EP-0570294-A1 2-Formylpyridine thiosemicarbazone derivatives, their preparation and their use as antitumor agents YALE UNIVERSITY (US) 1993-11-18 EP disclosed