SCHEMBL8688570

SCHEMBL8688570

CCN(C)c1ccc(-c2cc(C(F)(F)F)nn2-c2ccccc2S(N)(=O)=O)cc1F

nearest known ligand 0.58

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 15/20 0.58
PTGS1 P23219 5/20 0.58
PDPK1 O15530 4/20 0.45
F2 P00734 1/20 0.43
F10 P00742 1/20 0.43
KLKB1 P03952 1/20 0.43
PROC P04070 1/20 0.43
PRSS1 P07477 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8732522 0.92 PTGS2 (0.56) PTGS2PTGS1PDPK1F2F10
SCHEMBL8733795 0.91 PTGS2 (0.48) PTGS2PTGS1PDPK1
SCHEMBL8691417 0.91 PTGS2 (0.70) PTGS2PTGS1PDPK1
SCHEMBL8692115 0.90 PTGS2 (0.49) PTGS2PTGS1PDPK1
SCHEMBL8689252 0.87 PTGS2 (0.55) PTGS2PTGS1PDPK1
SCHEMBL8688939 0.85 PTGS2 (0.51) PTGS2PTGS1PDPK1
SCHEMBL8693453 0.84 PTGS2 (0.47) PTGS2PTGS1PDPK1
SCHEMBL6341483 0.84 PTGS2 (0.81) PTGS2PTGS1PDPK1
SCHEMBL8693370 0.83 PTGS2 (0.56) PTGS2PTGS1PDPK1
SCHEMBL8730016 0.82 PTGS2 (0.56) PTGS2PTGS1PDPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5760068-A NONSTEROIDAL ANTIINFLAMMATORY AGENTS WITH REDUCED SIDE EFFECTS G.D. SEARLE & CO. (US) 1998-06-02 US disclosed
US-5756529-A ANTIINFLAMMATORY G.D. SEARLE & CO. (US) 1998-05-26 US disclosed