SCHEMBL8689183

SCHEMBL8689183

COc1c(-c2cnc[nH]2)cccc1N(C)C1CCCC1

nearest known ligand 0.43

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 14/20 0.43
ADRA2A P08913 1/20 0.35
ADRA2B P18089 1/20 0.35
JAK2 O60674 1/20 0.35
JAK1 P23458 1/20 0.35
JAK3 P52333 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8687999 0.78 IDO1 (0.42) IDO1ADRA2AADRA2B
SCHEMBL8689417 0.78 IDO1 (0.43) IDO1ADRA2AADRA2B
SCHEMBL8687758 0.76 IDO1 (0.39) IDO1ADRA2AADRA2B
SCHEMBL8687672 0.75 IDO1 (0.48) IDO1ADRA2AADRA2B
SCHEMBL8687570 0.75 IDO1 (0.45) IDO1ADRA2AADRA2B
SCHEMBL8689303 0.74 IDO1 (0.47) IDO1ADRA2AADRA2B
SCHEMBL8687574 0.73 CYP1A2 (0.40) IDO1ADRA2AADRA2B
SCHEMBL24026598 0.72 IDO1 (0.65) IDO1ADRA2AADRA2B
SCHEMBL1241825 0.72 HPGD (0.40) ADRA2AADRA2BJAK2JAK1JAK3
SCHEMBL4065993 0.71 ADRA2A (0.50) IDO1ADRA2AADRA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5807860-A ACYLCOENZYME A:CHOLESTEROL ACYLTRANSFERASE INHIBITORS; HYPERLIPEMIA, ATHEROSCLEROSIS; ANTICHOLESTEROL AGENTS MITSUBISHI CHEMICAL CORPORATION (JP) 1998-09-15 US disclosed
EP-0773218-A1 N-(Piperazinylalkoxyphenyl)-N'phenylalkylurea derivatives as ACAT inhibitors for the treatment of atheroschlerosis MITSUBISHI CHEMICAL CORPORATION (JP) 1997-05-14 EP disclosed