SCHEMBL8692201

SCHEMBL8692201

COc1ccc(-c2c(Cl)cnn2-c2ccccc2S(N)(=O)=O)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 3/20 0.49
KDM4E B2RXH2 1/20 0.49
GAA P10253 1/20 0.49
PTGS2 P35354 2/20 0.49
PTGS1 P23219 1/20 0.49
NPSR1 Q6W5P4 2/20 0.48
ALDH1A1 P00352 2/20 0.48
LMNA P02545 1/20 0.48
NPBWR1 P48145 9/20 0.45
MCHR1 Q99705 4/20 0.43
SMN1; SMN2 Q16637 3/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
NPC1 O15118 1/20 0.41
S1PR4 O95977 1/20 0.41
MAPT P10636 1/20 0.41
S1PR1 P21453 1/20 0.41
RAB9A P51151 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8689437 0.87 HTT (0.49) HTTKDM4EGAAPTGS2PTGS1
SCHEMBL8689254 0.87 PTGS2 (0.52) PTGS2PTGS1NPSR1ALDH1A1LMNA
SCHEMBL8639255 0.87 PTGS2 (0.54) HTTKDM4EGAAPTGS2PTGS1
SCHEMBL7059925 0.86 PTGS2 (0.64) HTTPTGS2PTGS1NPSR1ALDH1A1
SCHEMBL8693825 0.86 PTGS2 (0.46) GAAPTGS2PTGS1ALDH1A1NPBWR1
SCHEMBL8691904 0.85 PTGS2 (0.49) PTGS2PTGS1CA12CA1CA2
SCHEMBL8693265 0.84 PTGS2 (0.52) PTGS2PTGS1NPSR1LMNAF10
SCHEMBL8691138 0.83 PTGS2 (0.50) HTTKDM4EGAAPTGS2PTGS1
SCHEMBL8688908 0.82 PTGS2 (0.43) GAAPTGS2PTGS1CA12CA1
SCHEMBL6343036 0.79 PTGS2 (0.71) HTTKDM4EGAAPTGS2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5760068-A NONSTEROIDAL ANTIINFLAMMATORY AGENTS WITH REDUCED SIDE EFFECTS G.D. SEARLE & CO. (US) 1998-06-02 US claimed
US-5760068-A NONSTEROIDAL ANTIINFLAMMATORY AGENTS WITH REDUCED SIDE EFFECTS G.D. SEARLE & CO. (US) 1998-06-02 US disclosed
US-5756529-A ANTIINFLAMMATORY G.D. SEARLE & CO. (US) 1998-05-26 US disclosed