SCHEMBL8699550

SCHEMBL8699550

c1ccc2c(c1)CC(Cc1nnn[nH]1)C2

nearest known ligand 0.46

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 3/20 0.46
IDO1 P14902 3/20 0.39
ADRA2A P08913 1/20 0.38
SIGMAR1 Q99720 2/20 0.33
PNMT P11086 2/20 0.32
HTR1A P08908 1/20 0.31
GRIN2B Q13224 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8700156 0.83 IDO1 (0.44) CYP19A1IDO1ADRA2ASIGMAR1PNMT
SCHEMBL8703698 0.76 PNMT (0.45) ADRA2APNMT
SCHEMBL6612499 0.75
SCHEMBL8703784 0.74 HTR2C (0.40) ADRA2AHTR1A
SCHEMBL3263413 0.72 PRCP (0.60)
SCHEMBL3940833 0.71 HRH4 (0.38)
SCHEMBL25010764 0.69
SCHEMBL6476895 0.69
SCHEMBL13406456 0.69 GBA1 (0.40)
SCHEMBL15721229 0.69 HRH3 (0.44)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998005651-A1 NOVEL GLUTAMATE RECEPTOR ANTAGONISTS: FUSED CYCLOALKYL QUINOXALINEDIONES WARNER-LAMBERT COMPANY (US) 1998-02-12 WO disclosed