SCHEMBL8700216

SCHEMBL8700216

CCCn1cnc2c1c(=O)n(CCCC(C)O)c(=O)n2C

nearest known ligand 0.69

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 8/20 0.68
LMNA P02545 2/20 0.68
ESR1 P03372 1/20 0.68
CYP1A2 P05177 1/20 0.68
MAPT P10636 1/20 0.68
NFKB1 P19838 1/20 0.68
ACHE P22303 1/20 0.68
BLM P54132 1/20 0.68
PMP22 Q01453 1/20 0.68
PDE4B Q07343 7/20 0.57
PDE4C Q08493 7/20 0.57
PDE4D Q08499 7/20 0.57
ADORA2A P29274 4/20 0.57
ADORA2B P29275 3/20 0.57
SMN1; SMN2 Q16637 1/20 0.55
TRPA1 O75762 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8702218 1.00 PDE4A (0.68) PDE4ALMNAESR1CYP1A2MAPT
SCHEMBL8695792 1.00 PDE4A (0.68) PDE4ALMNAESR1CYP1A2MAPT
SCHEMBL7989435 0.96 PDE4A (0.70) PDE4ALMNAESR1CYP1A2MAPT
SCHEMBL5256903 0.96 PDE4A (0.70) PDE4ALMNAESR1CYP1A2MAPT
SCHEMBL8697424 0.96 PDE4A (0.70) PDE4ALMNAESR1CYP1A2MAPT
SCHEMBL11612265 0.92 PDE4A (0.64) PDE4ALMNAESR1CYP1A2MAPT
SCHEMBL4345194 0.92 PDE4A (0.64) PDE4ALMNAESR1CYP1A2MAPT
SCHEMBL10788514 0.91 PDE4A (0.62) PDE4ALMNAESR1CYP1A2MAPT
SCHEMBL11611955 0.91 PDE4A (0.62) PDE4ALMNAESR1CYP1A2MAPT
SCHEMBL11614003 0.91 PDE4A (0.62) PDE4ALMNAESR1CYP1A2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5710272-A INCREASING CEREBRAL BLOOD FLOW HOECHST AKTIENGESELLSCHAFT (DE) 1998-01-20 US disclosed
EP-0435152-B1 Process for the enantioselective preparation of (omega-1)-hydroxyalkylxanthines HOECHST AG (DE) 1996-11-13 EP disclosed
US-5472873-A Rhodotorula rubra useful in a process for the preparation of (ω-1)-hydroxyalkylxanthines HOECHST AKTIENGESELLSCHAFT (DE) 1995-12-05 US disclosed
US-5310666-A Vascular disorders HOECHST AKTIENGESELLSCHAFT (DE) 1994-05-10 US disclosed
EP-0435152-A2 Process for the enantioselective preparation of (omega-1)-hydroxyalkylxanthines HOECHST AKTIENGESELLSCHAFT (DE) 1991-07-03 EP disclosed