SCHEMBL8700941

SCHEMBL8700941

Brc1ccc(-c2cnccn2)cc1.[Li]CCCC

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 5/20 0.60
CYP19A1 P11511 3/20 0.60
CYP2C9 P11712 3/20 0.60
CYP2C19 P33261 3/20 0.60
NPC1 O15118 3/20 0.48
RAB9A P51151 3/20 0.48
L3MBTL1 Q9Y468 2/20 0.48
SMN1; SMN2 Q16637 2/20 0.48
NFKB1 P19838 1/20 0.48
MAPK1 P28482 1/20 0.48
NFKB2 Q00653 1/20 0.48
RELA Q04206 1/20 0.48
TERT O14746 2/20 0.38
BRS3 P32247 1/20 0.38
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 2/20 0.36
SREBF2 Q12772 1/20 0.35
KDM4E B2RXH2 1/20 0.34
LMNA P02545 1/20 0.34
MAPT P10636 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL999538 0.82 CYP19A1 (0.51) CYP2D6CYP19A1CYP2C9CYP2C19NPC1
SCHEMBL8695286 0.79 CYP2D6 (0.60) CYP2D6CYP19A1CYP2C9CYP2C19NPC1
SCHEMBL21984930 0.76 CYP2D6 (0.55) CYP2D6CYP19A1CYP2C9CYP2C19NPC1
SCHEMBL14129889 0.75 CYP2D6 (1.00) CYP2D6CYP19A1CYP2C9CYP2C19NPC1
SCHEMBL11541937 0.73 CYP2D6 (0.60) CYP2D6CYP19A1CYP2C9CYP2C19NPC1
SCHEMBL9777426 0.73 CYP2D6 (0.63) CYP2D6CYP19A1CYP2C9CYP2C19NPC1
SCHEMBL8957199 0.72 CYP2D6 (0.91) CYP2D6CYP19A1CYP2C9CYP2C19NPC1
SCHEMBL1109087 0.71 CYP2D6 (0.56) CYP2D6CYP19A1CYP2C9CYP2C19NPC1
SCHEMBL31140236 0.71 CYP2D6 (0.56) CYP2D6CYP19A1CYP2C9CYP2C19NPC1
SCHEMBL31140242 0.71 CYP2D6 (0.61) CYP2D6CYP19A1CYP2C9CYP2C19NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998004260-A1 SUBSTITUTED BIPHENYL SULFONAMIDE ENDOTHELIN ANTAGONISTS BRISTOL-MYERS SQUIBB COMPANY (US) 1998-02-05 WO disclosed