SCHEMBL8701044

SCHEMBL8701044

CCc1cc(NC(=S)N2CCN(c3ccccc3F)CC2)c(OC)nc1C

nearest known ligand 0.65

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 5/20 0.65
ATM Q13315 2/20 0.65
PKM P14618 1/20 0.56
ALDH1A1 P00352 4/20 0.55
KDM4E B2RXH2 3/20 0.55
HTT P42858 2/20 0.48
GAA P10253 1/20 0.48
MAPT P10636 1/20 0.48
RAB9A P51151 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
MEN1 O00255 2/20 0.48
LMNA P02545 2/20 0.46
NPSR1 Q6W5P4 2/20 0.46
TSHR P16473 1/20 0.46
PHGDH O43175 1/20 0.46
CYP1A2 P05177 1/20 0.45
CYP2C9 P11712 1/20 0.45
CYP2C19 P33261 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6653829 0.92 KMT2A (0.55) KMT2AATMPKMALDH1A1KDM4E
SCHEMBL6652670 0.90 PHGDH (0.58) KMT2AATMALDH1A1KDM4EGAA
SCHEMBL8704636 0.90 KMT2A (0.57) KMT2AATMALDH1A1KDM4EMAPT
SCHEMBL6657797 0.87 KMT2A (0.48) KMT2AATMPKMALDH1A1KDM4E
SCHEMBL6652409 0.87 KMT2A (0.48) KMT2AATMPKMALDH1A1GAA
SCHEMBL6651274 0.86 MEN1 (0.54) KMT2AALDH1A1GAAMAPTSMN1; SMN2
SCHEMBL8699351 0.84 ALDH1A1 (0.66) KMT2AALDH1A1KDM4EHTTGAA
SCHEMBL6654791 0.83 PHGDH (0.43) KMT2AATMALDH1A1KDM4EMAPT
SCHEMBL6657804 0.83 SMN1; SMN2 (0.46) KMT2AATMALDH1A1MAPTSMN1; SMN2
SCHEMBL6653052 0.82 PHGDH (0.56) KMT2APKMALDH1A1GAAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5780472-A ANTITUMOR AGENTS SAMJIN PHARMACEUTICAZL CO., LTD. (KR) 1998-07-14 US disclosed
WO-1996021648-A1 NEW PIPERAZINE DERIVATIVES AND METHODS FOR THE PREPARATION THEREOF AND COMPOSITIONS CONTAINING THE SAME SAMJIN PHARMACEUTICAL CO., LTD. (KR) 1996-07-18 WO disclosed