SCHEMBL8701190

SCHEMBL8701190

CCN1c2ncccc2C(=O)N(C)c2ccc(-c3c[nH]nc3C)nc21

nearest known ligand 0.42

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.42
CYP2C9 P11712 2/20 0.42
CYP2C19 P33261 2/20 0.42
CYP1A2 P05177 1/20 0.37
BRD4 O60885 17/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8546643 0.82 CYP3A4 (0.42) CYP3A4CYP2C9CYP2C19CYP1A2BRD4
SCHEMBL8547631 0.81 CYP3A4 (0.39) CYP3A4CYP2C9CYP2C19CYP1A2BRD4
SCHEMBL8702103 0.80 SIRT2 (0.43) CYP3A4CYP2C9CYP2C19BRD4
SCHEMBL8701364 0.79 CYP3A4 (0.39) CYP3A4CYP2C9CYP2C19CYP1A2BRD4
SCHEMBL8545648 0.79 CYP3A4 (0.39) CYP3A4CYP2C9CYP2C19CYP1A2BRD4
SCHEMBL8300415 0.78 CYP3A4 (0.45) CYP3A4CYP2C9CYP2C19CYP1A2BRD4
SCHEMBL8299587 0.78 CYP3A4 (0.52) CYP3A4CYP2C9CYP2C19BRD4
SCHEMBL8701079 0.78 CYP3A4 (0.39) CYP3A4CYP2C9CYP2C19CYP1A2BRD4
SCHEMBL8306273 0.78 CYP3A4 (0.44) CYP3A4CYP2C9CYP2C19CYP1A2BRD4
SCHEMBL8889357 0.78 CYP3A4 (0.42) CYP3A4CYP2C9CYP2C19CYP1A2BRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5837704-A PREVENTION OR TREATMENT OF AIDS BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 1998-11-17 US disclosed