SCHEMBL8702103

SCHEMBL8702103

CCN1c2ncccc2C(=O)N(C)c2ccc(-c3c[nH]c4ccccc34)nc21

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIRT2 Q8IXJ6 2/20 0.43
SIRT1 Q96EB6 1/20 0.43
GSK3B P49841 2/20 0.41
CLK1 P49759 1/20 0.41
CDK5 Q00535 1/20 0.41
DYRK1A Q13627 1/20 0.41
CDK5R1 Q15078 1/20 0.41
MAP3K14 Q99558 1/20 0.41
PIM1 P11309 1/20 0.41
BRD4 O60885 2/20 0.41
CDK1 P06493 1/20 0.40
CCNB1 P14635 1/20 0.40
PDGFRB P09619 3/20 0.39
EIF2AK2 P19525 1/20 0.38
MAPT P10636 3/20 0.38
CDK2 P24941 2/20 0.38
MEN1 O00255 1/20 0.38
NPC1 O15118 1/20 0.38
GAA P10253 1/20 0.38
RAB9A P51151 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8701190 0.80 CYP3A4 (0.42) BRD4CYP3A4CYP2C9CYP2C19
SCHEMBL8547631 0.80 CYP3A4 (0.39) BRD4CYP3A4CYP2C9CYP2C19
SCHEMBL8545648 0.80 CYP3A4 (0.39) BRD4CYP3A4CYP2C9CYP2C19
SCHEMBL8707904 0.78 BRD4 (0.39) BRD4CYP3A4CYP2C9CYP2C19
SCHEMBL8546643 0.78 CYP3A4 (0.42) CLK1BRD4MAPK8CYP3A4CYP2C9
SCHEMBL8701057 0.78 CYP3A4 (0.40) BRD4CYP3A4CYP2C9CYP2C19
SCHEMBL8701364 0.78 CYP3A4 (0.39) BRD4CYP3A4CYP2C9CYP2C19
SCHEMBL8299587 0.77 CYP3A4 (0.52) BRD4CYP3A4CYP2C9CYP2C19ALDH1A1
SCHEMBL8701079 0.77 CYP3A4 (0.39) BRD4CYP3A4CYP2C9CYP2C19
SCHEMBL8306273 0.77 CYP3A4 (0.44) BRD4CYP3A4CYP2C9CYP2C19ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5837704-A PREVENTION OR TREATMENT OF AIDS BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 1998-11-17 US disclosed