SCHEMBL8701939

SCHEMBL8701939

CN(c1ccc(OC(F)(F)F)c(CC2(c3ccccc3)CCCCN2N)c1)S(C)(=O)=O

nearest known ligand 0.35

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 2/20 0.35
DRD2 P14416 4/20 0.35
SLC6A3 Q01959 4/20 0.35
OPRD1 P41143 1/20 0.33
OPRK1 P41145 1/20 0.33
PTGDR2 Q9Y5Y4 4/20 0.33
SLC6A2 P23975 1/20 0.32
PTGS2 P35354 1/20 0.32
PTK2 Q05397 1/20 0.31
BRD4 O60885 1/20 0.31
NR1I2 O75469 1/20 0.31
RORC P51449 1/20 0.31
OPRL1 P41146 2/20 0.31
ABL1 P00519 2/20 0.31
CYP19A1 P11511 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8707886 0.99 TACR1 (0.35) TACR1DRD2SLC6A3OPRD1OPRK1
SCHEMBL8706170 0.92 DRD2 (0.34) TACR1DRD2SLC6A3OPRD1OPRK1
Hydrochloric Acid SCHEMBL8706566 0.91 DRD2 (0.33) TACR1DRD2SLC6A3OPRD1OPRK1
SCHEMBL8701385 0.89 TACR1 (0.45) TACR1PTGS2
SCHEMBL8701299 0.86 TACR1 (0.36) TACR1PTGS2BRD4CYP19A1
Hydrochloric Acid SCHEMBL8702143 0.86 TACR1 (0.35) TACR1PTGS2BRD4CYP19A1
SCHEMBL8707766 0.85 TACR1 (0.38) TACR1SLC6A2CYP19A1
SCHEMBL8705094 0.84 TACR1 (0.35) TACR1RORCOPRL1
Hydrochloric Acid SCHEMBL8707618 0.83 TACR1 (0.37) TACR1CYP19A1
Hydrochloric Acid SCHEMBL8706672 0.83 TACR1 (0.35) TACR1RORCOPRL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5721255-A Substituted benzylamino nitrogen containing non-aromatic heterocycles PFIZER INC. (US) 1998-02-24 US claimed
US-5721255-A Substituted benzylamino nitrogen containing non-aromatic heterocycles PFIZER INC. (US) 1998-02-24 US disclosed