SCHEMBL8703231

SCHEMBL8703231

COc1cccc(CCc2ccccc2OC[C@@H]2CCCN2)c1

nearest known ligand 0.63

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ABCB1 P08183 13/20 0.60
HTR1A P08908 4/20 0.60
DRD2 P14416 4/20 0.60
CHRNB4 P30926 1/20 0.59
CHRNA3 P32297 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8703238 1.00 ABCB1 (0.60) ABCB1HTR1ADRD2CHRNB4CHRNA3
Hydrochloric Acid SCHEMBL8703399 0.99 ABCB1 (0.59) ABCB1HTR1ADRD2CHRNB4CHRNA3
Hydrochloric Acid SCHEMBL8703779 0.99 ABCB1 (0.59) ABCB1HTR1ADRD2CHRNB4CHRNA3
Hydrochloric Acid SCHEMBL8703392 0.99 ABCB1 (0.59) ABCB1HTR1ADRD2CHRNB4CHRNA3
SCHEMBL21095169 0.86 ABCB1 (0.59) ABCB1HTR1ADRD2
SCHEMBL21095600 0.86 ABCB1 (0.59) ABCB1HTR1ADRD2
SCHEMBL21095171 0.86 ABCB1 (0.59) ABCB1HTR1ADRD2
Hydrochloric Acid SCHEMBL8702021 0.85 TP53 (0.57) ABCB1HTR1ADRD2
SCHEMBL27341184 0.85 CHRNB4 (0.60) HTR1ADRD2CHRNB4CHRNA3
Hydrochloric Acid SCHEMBL8707931 0.84 CHRNB4 (0.59) HTR1ADRD2CHRNB4CHRNA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0844000-A1 Use of alpha, omega-diarylalkane derivatives in the treatment and prevention of psychosis SANKYO COMPANY LIMITED (JP) 1998-05-27 EP disclosed
US-5556864-A TREATMENT OF CIRCULATORY DISEASES AND PSYCHOSIS SANKYO COMPANY, LIMITED (JP) 1996-09-17 US disclosed
EP-0600717-A1 Phenoxyalkylamines, -pyrrolidines and -piperidines for the treatment and prevention of circulatory diseases and psychosis SANKYO COMPANY LIMITED (JP) 1994-06-08 EP disclosed