SCHEMBL8708223

SCHEMBL8708223

O=C(NCC1(Cc2ccccc2)CCN(Cc2ccccc2)CC1)N1CCOCC1

nearest known ligand 0.60

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
NPFFR1 Q9GZQ6 17/20 0.60
NPFFR2 Q9Y5X5 17/20 0.60
OPRK1 P41145 2/20 0.59
ALDH1A1 P00352 1/20 0.49
OPRM1 P35372 1/20 0.47
OPRD1 P41143 1/20 0.47
NPC1 O15118 1/20 0.46
HTT P42858 1/20 0.46
RAB9A P51151 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8709388 0.85 HTT (0.46) NPFFR1NPFFR2OPRK1ALDH1A1OPRM1
SCHEMBL8707282 0.77 CYP2D6 (0.50) ALDH1A1NPC1HTTRAB9ASMN1; SMN2
SCHEMBL20572136 0.74 NPFFR1 (0.60) NPFFR1NPFFR2OPRK1ALDH1A1OPRM1
SCHEMBL4630062 0.73 NPFFR1 (0.58) NPFFR1NPFFR2OPRK1ALDH1A1
SCHEMBL8393626 0.73 USP2 (0.64) ALDH1A1HTT
SCHEMBL4631287 0.73 NPFFR1 (0.57) NPFFR1NPFFR2OPRK1ALDH1A1
SCHEMBL8708218 0.73 ALDH1A1 (0.48) ALDH1A1NPC1HTTRAB9ASMN1; SMN2
SCHEMBL12195395 0.73 NPFFR1 (0.58) NPFFR1NPFFR2OPRK1ALDH1A1
SCHEMBL16915597 0.72 NPFFR1 (0.57) NPFFR1NPFFR2OPRK1ALDH1A1OPRM1
SCHEMBL5995214 0.72 POLB (0.77) ALDH1A1OPRM1OPRD1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1998018762-A1 NEW DERIVATIVES OF DIVERSELY SUBSTITUTED CYCLICAL AMIDE SELECTIVE ANTAGONISTS OF THE HUMAN RECEPTOR NK3, PROCESS FOR OBTAINING THEM, AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM SANOFI (FR) 1998-05-07 WO disclosed