SCHEMBL8710107

SCHEMBL8710107

CCCn1c(=O)c2[nH]c(C(C)Cc3ccc(O)cc3)nc2n(CCC)c1=O

nearest known ligand 0.80

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
ADORA2B P29275 3/20 0.65
ADORA2A P29274 2/20 0.65

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8706990 0.89 KDM4E (0.63) ADORA2BADORA2A
SCHEMBL721663 0.89 KDM4E (0.63) ADORA2BADORA2A
SCHEMBL194851 0.89 KDM4E (0.63) ADORA2BADORA2A
SCHEMBL7269136 0.88
SCHEMBL8713814 0.84 ADORA2B (0.57) ADORA2B
SCHEMBL10675262 0.81 ADORA2A (0.66) ADORA2BADORA2A
SCHEMBL8709837 0.80 ADORA2B (0.61) ADORA2BADORA2A
SCHEMBL1948455 0.79 ADORA2B (1.00) ADORA2BADORA2A
SCHEMBL8705703 0.77
SCHEMBL8705440 0.76

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1041418-C Xanthine derivatives as adenosine A1 receptor antagonists MERRELL DOW PHARMA (US) 1998-12-30 CN claimed
US-5047534-A Xanthine derivatives; hyupotensive agents, cardiotonic agents MERRELL DOW PHARMACEUTICALS INC. (US) 1991-09-10 US claimed
CN-1041418-C Xanthine derivatives as adenosine A1 receptor antagonists MERRELL DOW PHARMA (US) 1998-12-30 CN disclosed
US-5840729-A ATTENUATING COGNITIVE DEFICIT MERRELL PHARMACEUTICALS INC. (US) 1998-11-24 US disclosed
EP-0686155-A1 XANTHINE DERIVATIVES AS ADENOSINE A1 RECEPTOR ANTAGONISTS MERRELL PHARMACEUTICALS INC. (US) 1995-12-13 EP disclosed
WO-1994019349-A1 XANTHINE DERIVATIVES AS ADENOSINE A1 RECEPTOR ANTAGONISTS MERRELL DOW PHARMACEUTICALS INC. (US) 1994-09-01 WO disclosed
US-5047534-A Xanthine derivatives; hyupotensive agents, cardiotonic agents MERRELL DOW PHARMACEUTICALS INC. (US) 1991-09-10 US disclosed