SCHEMBL8713451

SCHEMBL8713451

CC(C)(C)ON=C(c1cc(C(F)(F)F)ccc1O)c1ncccc1C#N

nearest known ligand 0.35

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ELANE P08246 2/20 0.34
TLR7 Q9NYK1 2/20 0.33
KDM4E B2RXH2 2/20 0.32
CYP1A2 P05177 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
RECQL P46063 1/20 0.32
TAS2R14 Q9NYV8 1/20 0.31
COMT P21964 1/20 0.31
TRPV1 Q8NER1 1/20 0.31
GAA P10253 1/20 0.31
CNR2 P34972 1/20 0.30
TBXA2R P21731 2/20 0.30
L3MBTL1 Q9Y468 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8713450 1.00 ELANE (0.34) ELANETLR7KDM4ECYP1A2CYP2C9
SCHEMBL8709612 0.87 TLR7 (0.42) TLR7KDM4ECOMTGAATBXA2R
SCHEMBL8709608 0.87 TLR7 (0.42) TLR7KDM4ECOMTGAATBXA2R
SCHEMBL8715533 0.86 MAPT (0.37) ELANEKDM4ERECQLL3MBTL1
SCHEMBL8712087 0.86 KDM4C (0.32)
SCHEMBL8715532 0.86 MAPT (0.37) ELANEKDM4ERECQLL3MBTL1
SCHEMBL8715196 0.86 KDM4C (0.32)
SCHEMBL8709848 0.86 TLR7 (0.36) TLR7
SCHEMBL8709849 0.86 TLR7 (0.36) TLR7
SCHEMBL8710689 0.85 MEN1 (0.35) KDM4EGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5716971-A FOR TREATMENT OF ANGINA PECTORIS AND HYPERTENSION TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-02-10 US disclosed
EP-0623597-B1 Pyridine derivatives, with potassium channel opening activity TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1997-10-22 EP disclosed
EP-0623597-A1 Pyridine derivatives, with potassium channel opening activity Takeda Chemical Industries, Ltd. (JP) 1994-11-09 EP disclosed