SCHEMBL8713946

SCHEMBL8713946

CN1C2COCC1CC(NC(=O)c1n[nH]c3ccccc13)C2

nearest known ligand 0.83

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.61
RAB9A P51151 1/20 0.61
HTR3A P46098 11/20 0.57
GSK3B P49841 1/20 0.55
DYRK1A Q13627 1/20 0.55
RIPK1 Q13546 1/20 0.54
SMYD3 Q9H7B4 1/20 0.54
USP30 Q70CQ3 1/20 0.53
YTHDC1 Q96MU7 1/20 0.52
CHRNA7 P36544 1/20 0.52
ALDH1A1 P00352 1/20 0.52
CYP3A4 P08684 1/20 0.52
TSHR P16473 1/20 0.52
MAPK1 P28482 1/20 0.52
HSD17B10 Q99714 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8713942 1.00 NPC1 (0.61) NPC1RAB9AHTR3AGSK3BDYRK1A
SCHEMBL2086084 0.91 NPC1 (0.67) NPC1RAB9AHTR3AGSK3BDYRK1A
SCHEMBL8719122 0.90 NPC1 (0.58) NPC1RAB9AHTR3AGSK3BDYRK1A
SCHEMBL8714813 0.89 NPC1 (0.57) NPC1RAB9AHTR3AGSK3BDYRK1A
SCHEMBL8714762 0.89 NPC1 (0.57) NPC1RAB9AHTR3AGSK3BDYRK1A
SCHEMBL12441936 0.89 NPC1 (0.68) NPC1RAB9AHTR3AGSK3BDYRK1A
SCHEMBL7345995 0.89 NPC1 (0.61) NPC1RAB9AHTR3AGSK3BDYRK1A
Indisetron SCHEMBL332330 0.89 NPC1 (0.61) NPC1RAB9AHTR3AGSK3BDYRK1A
SCHEMBL2087490 0.89 NPC1 (0.68) NPC1RAB9AHTR3AGSK3BDYRK1A
SCHEMBL2086948 0.89 NPC1 (0.68) NPC1RAB9AHTR3AGSK3BDYRK1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0708105-B1 5-HT4 receptor agonists NISSHIN FLOUR MILLING CO (JP) 1998-12-23 EP disclosed
EP-0708105-A1 5-HT4 receptor agonists NISSHIN FLOUR MILLING CO., LTD. (JP) 1996-04-24 EP disclosed