SCHEMBL8714827

SCHEMBL8714827

Cc1cn(Nc2ccncc2)c2ccc(O)cc12.Cc1cn(Nc2ccncc2)c2ccc(OCc3ccccc3)cc12

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 2/20 0.53
F2 P00734 2/20 0.46
KCNH2 Q12809 1/20 0.44
GRIN2B Q13224 1/20 0.44
EGFR P00533 1/20 0.41
ERBB2 P04626 1/20 0.41
BCHE P06276 1/20 0.41
ACHE P22303 1/20 0.41
MEN1 O00255 4/20 0.41
KMT2A Q03164 4/20 0.41
RAB9A P51151 3/20 0.41
NPC1 O15118 2/20 0.41
GAA P10253 3/20 0.40
MAPT P10636 3/20 0.40
MAOB P27338 3/20 0.40
PKM P14618 3/20 0.40
BLM P54132 2/20 0.40
ALDH1A1 P00352 2/20 0.40
L3MBTL1 Q9Y468 2/20 0.40
THRB P10828 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7608007 0.95 SLC6A2 (0.58) SLC6A2F2KCNH2GRIN2BBCHE
SCHEMBL7613199 0.84 SLC6A2 (0.65) SLC6A2BCHEACHEGAADYRK1A
SCHEMBL8539866 0.79 BCHE (0.63) SLC6A2F2KCNH2GRIN2BBCHE
SCHEMBL10336609 0.79 SLC6A2 (0.52) SLC6A2EGFRMEN1KMT2AGAA
SCHEMBL8539616 0.74 SLC6A2 (0.56) SLC6A2F2KCNH2GRIN2BMEN1
SCHEMBL7620289 0.73 BCHE (0.45) F2KCNH2GRIN2BBCHEACHE
SCHEMBL8836224 0.73 SPHK2 (0.48) MEN1KMT2ARAB9ANPC1MAOB
SCHEMBL8836219 0.73 LTA4H (0.50) MEN1KMT2ARAB9ANPC1MAOB
SCHEMBL7620284 0.72 BCHE (0.43) F2KCNH2GRIN2BBCHEACHE
SCHEMBL8544882 0.72 NPC1 (0.53) MEN1KMT2ARAB9ANPC1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0840609-A1 USE OF UNSUBSTITUTED AND SUBSTITUTED N-(PYRROL-1-YL)PYRIDINAMINES AS ANTICONVULSANT AGENTS HOECHST MARION ROUSSEL, INC. (US) 1998-05-13 EP disclosed
WO-1997004777-A1 USE OFF UNSUBSTITUTED AND SUBSTITUTED N-(PYRROL-1-YL)PYRIDINAMINES AS ANTICONVULSANT AGENTS HOECHST MARION ROUSSEL, INC. (US) 1997-02-13 WO disclosed