SCHEMBL8715325

SCHEMBL8715325

COc1ccc(-c2ccc(CN)cc2)cc1C(=O)NC1CCC(C(=O)O)CC1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 1/20 0.49
NR1H4 Q96RI1 1/20 0.46
CNR1 P21554 10/20 0.45
CNR2 P34972 10/20 0.45
TAS1R3 Q7RTX0 1/20 0.45
TAS1R1 Q7RTX1 1/20 0.45
TAS1R2 Q8TE23 1/20 0.45
L3MBTL1 Q9Y468 2/20 0.45
PRSS1 P07477 1/20 0.44
PRSS2 P07478 1/20 0.44
PRSS3 P35030 1/20 0.44
ST14 Q9Y5Y6 1/20 0.44
ALDH1A1 P00352 2/20 0.44
KDM4E B2RXH2 1/20 0.43
LMNA P02545 1/20 0.43
POLB P06746 1/20 0.43
MAPT P10636 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
ADRA2A P08913 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8715395 0.92 KDM1A (0.47) KDM1ANR1H4CNR1CNR2TAS1R3
SCHEMBL8410563 0.84 KDM1A (0.48) KDM1ACNR1CNR2PRSS1PRSS2
SCHEMBL8407420 0.79 NPC1 (0.53) PRSS1PRSS2PRSS3ST14DRD2
SCHEMBL8410171 0.76 CFTR (0.48) KDM1AL3MBTL1PRSS1PRSS2PRSS3
SCHEMBL8410733 0.74 POLB (0.55) NR1H4ALDH1A1POLB
SCHEMBL8407182 0.74 SMYD3 (0.49) PRSS1PRSS2PRSS3ST14DRD2
Hydrochloric Acid SCHEMBL8949029 0.73 CNR2 (0.49) CNR1CNR2RAB9A
Hydrochloric Acid SCHEMBL4733281 0.72 PDE4B (0.50) KDM1AL3MBTL1ALDH1A1KDM4ELMNA
SCHEMBL21482092 0.72 NAAA (0.43) CNR1CNR2POLBDRD3KCNH2
SCHEMBL9568223 0.72 ST14 (0.40) KDM1APRSS1PRSS2PRSS3ST14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0496378-B1 Biphenylderivatives, drugs containing these compounds and processes for their preparation THOMAE GMBH DR K (DE) 1995-09-20 EP claimed
US-5736559-A CARDIOVASCULAR DISORDERS; RESPIRATORY SYSTEM DISORDERS KARL THOMAE GMBH (DE) 1998-04-07 US disclosed
US-5597825-A AGGREGATION INHIBITORS DR. KARL THOMAE GMBH (DE) 1997-01-28 US disclosed
EP-0496378-B1 Biphenylderivatives, drugs containing these compounds and processes for their preparation THOMAE GMBH DR K (DE) 1995-09-20 EP disclosed
EP-0496378-A1 Biphenylderivatives, drugs containing these compounds and processes for their preparation Dr. Karl Thomae GmbH (DE) 1992-07-29 EP disclosed