SCHEMBL8715328

SCHEMBL8715328

BrCCOC1c2ccccc2CCc2ccccc21

nearest known ligand 0.44

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
RET P07949 2/20 0.44
HTR2A P28223 1/20 0.44
CHRNA7 P36544 4/20 0.40
CHRNB2 P17787 2/20 0.40
CHRNA4 P43681 2/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
HIF1A Q16665 1/20 0.40
IDO1 P14902 2/20 0.38
ACP3 P15309 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8712643 0.81 RET (0.44) RETHTR2ACHRNA7CHRNB2CHRNA4
SCHEMBL6965256 0.80 MAPT (0.47) RETHTR2ACYP2D6
SCHEMBL19359221 0.79 IDO1 (0.56) RETHTR2AIDO1
SCHEMBL30729415 0.77 RET (0.66) RETHTR2ACYP2D6
SCHEMBL13447594 0.77 HTR2A (0.47) RETHTR2ACHRNA7CHRNB2CHRNA4
SCHEMBL7979437 0.76 HTR2A (0.47) RETHTR2ACHRNA7CHRNB2CHRNA4
SCHEMBL7965950 0.76 HTR2A (0.47) RETHTR2AIDO1
SCHEMBL7468970 0.74 KCNA3 (0.45) RETHTR2ACYP2D6
SCHEMBL9084723 0.74 KDM4E (0.38) RETHTR2ACHRNA7CHRNB2CHRNA4
SCHEMBL9084730 0.74 KDM4E (0.38) RETHTR2ACHRNA7CHRNB2CHRNA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0820442-A1 NOVEL HETEROCYCLIC COMPOUNDS NOVO NORDISK A/S (DK) 1998-01-28 EP disclosed
WO-1996031474-A1 NOVEL HETEROCYCLIC COMPOUNDS NOVO NORDISK A/S (DK) 1996-10-10 WO disclosed