SCHEMBL8715414

SCHEMBL8715414

COC(=O)c1ccccc1N(CCN1CCC(C(=O)c2ccc(F)cc2)CC1)C(=O)c1ccc(N)cc1

nearest known ligand 0.48

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CYP2D6 P10635 2/20 0.46
CYP2C19 P33261 1/20 0.46
HTR2A P28223 3/20 0.46
HSD11B1 P28845 2/20 0.46
KDM4E B2RXH2 1/20 0.46
CYP1A2 P05177 1/20 0.46
CYP3A4 P08684 1/20 0.46
LMNA P02545 1/20 0.46
KMT2A Q03164 1/20 0.46
HTR2C P28335 2/20 0.45
HTR7 P34969 2/20 0.45
HTR6 P50406 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8710975 0.89 KMT2A (0.48) CYP2D6CYP2C19HTR2AHSD11B1KDM4E
SCHEMBL8711071 0.89 CYP2D6 (0.52) CYP2D6CYP2C19HTR2AHSD11B1KDM4E
SCHEMBL8713822 0.88 HTR2A (0.51) CYP2D6CYP2C19HTR2AHSD11B1KDM4E
Fumaric Acid SCHEMBL8711175 0.85 SMN1; SMN2 (0.46) CYP2D6CYP2C19HTR2AKDM4ECYP1A2
Fumaric Acid SCHEMBL8711179 0.85 SMN1; SMN2 (0.46) CYP2D6CYP2C19HTR2AKDM4ECYP1A2
Fumaric Acid SCHEMBL9230570 0.84 CYP2D6 (0.48) CYP2D6CYP2C19HTR2AHSD11B1KDM4E
Fumaric Acid SCHEMBL9230577 0.84 CYP2D6 (0.48) CYP2D6CYP2C19HTR2AHSD11B1KDM4E
SCHEMBL9230053 0.83 HTR2A (0.48) CYP2D6CYP2C19HTR2AKDM4ECYP1A2
SCHEMBL8711222 0.83 HTR2A (0.48) CYP2D6HTR2AKDM4ECYP1A2CYP3A4
SCHEMBL8710869 0.82 ACHE (0.56) CYP2D6HTR2AKDM4ECYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5728835-A HYPOTENSIVE AGENTS; ANTIISCHEMIC AGENTS TOA EIYO, LTD. (JP) 1998-03-17 US disclosed
WO-1996034851-A1 BENZENE, PYRIDINE, NAPHTALENE OR BENZOPHENONE DERIVATIVES AS INHIBITORS OF SQUALENE SYNTHETASE AND PROTEIN FARNESYLTRANSFERASE ABBOTT LABORATORIES (US) 1996-11-07 WO disclosed
EP-0661266-A1 Substituted cyclic amine compounds as 5HT2 antagonists TOA EIYO LTD. (JP) 1995-07-05 EP disclosed