SCHEMBL8715705

SCHEMBL8715705

CC(CN)(Cc1c[nH]c2ccccc12)OC(=O)NC(CO)C(O)c1ccccc1

nearest known ligand 0.46

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 16/20 0.46
TACR3 P29371 1/20 0.46
CTSL P07711 1/20 0.44
CTSS P25774 1/20 0.44
CTSK P43235 1/20 0.44
ADRB3 P13945 1/20 0.42
SSTR3 P32745 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8705433 0.87 TACR1 (0.46) TACR1TACR3CTSLCTSSCTSK
SCHEMBL6888854 0.81 TACR1 (0.46) TACR1TACR3ADRB3
SCHEMBL9539175 0.81 ADRB3 (0.44) TACR1TACR3ADRB3
SCHEMBL8892928 0.78 TACR1 (0.57) TACR1TACR3
SCHEMBL9293320 0.77 TACR1 (0.45) TACR1TACR3ADRB3
SCHEMBL8894105 0.77 TACR1 (0.51) TACR1TACR3
SCHEMBL9293315 0.76 TACR1 (0.45) TACR1TACR3ADRB3
SCHEMBL8715712 0.76 TACR3 (0.50) TACR1TACR3ADRB3
SCHEMBL9293660 0.76 TACR1 (0.48) TACR1TACR3
SCHEMBL8893069 0.75 TACR1 (0.44) TACR1TACR3ADRB3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5726200-A Pro-drugs for CCK antagonists WARNER-LAMBERT COMPANY (US) 1998-03-10 US disclosed