SCHEMBL9539175

SCHEMBL9539175

CC(CNC(CO)C(O)c1ccccc1)(Cc1c[nH]c2ccccc12)OC(N)=O

nearest known ligand 0.44

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ADRB3 P13945 1/20 0.44
TACR1 P25103 14/20 0.44
TACR3 P29371 1/20 0.44
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
CYP2D6 P10635 1/20 0.41
MMP9 P14780 1/20 0.40
MMP8 P22894 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6888854 0.83 TACR1 (0.46) ADRB3TACR1TACR3MEN1KMT2A
SCHEMBL7669465 0.82 ADRB3 (0.44) ADRB3TACR1TACR3MEN1KMT2A
SCHEMBL8715705 0.81 TACR1 (0.46) ADRB3TACR1TACR3
SCHEMBL8705433 0.80 TACR1 (0.46) ADRB3TACR1TACR3MEN1KMT2A
SCHEMBL8705350 0.78 PKM (0.47) ADRB3TACR1MEN1KMT2ACYP2D6
SCHEMBL9293660 0.76 TACR1 (0.48) TACR1TACR3
SCHEMBL9538103 0.75 TACR1 (0.38) ADRB3TACR1TACR3MMP9MMP8
SCHEMBL8892928 0.74 TACR1 (0.57) TACR1TACR3
SCHEMBL8485370 0.74 TACR1 (0.61) TACR1TACR3MEN1KMT2A
SCHEMBL9274807 0.74 TACR1 (0.61) TACR1TACR3MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1993003721-A1 CHOLECYSTOKININ ANTAGONISTS USEFUL FOR TREATING DEPRESSION WARNER-LAMBERT COMPANY (US) 1993-03-04 WO claimed
WO-1993003721-A1 CHOLECYSTOKININ ANTAGONISTS USEFUL FOR TREATING DEPRESSION WARNER-LAMBERT COMPANY (US) 1993-03-04 WO disclosed
EP-0479910-A1 N-SUBSTITUTED CYCLOALKYL AND POLYCYCLOALKYL ALPHA-SUBSTITUTED Trp-Phe- AND PHENETHYLAMINE DERIVATIVES WARNER-LAMBERT COMPANY (US) 1992-04-15 EP disclosed
WO-1991000274-A1 N-SUBSTITUTED CYCLOALKYL AND POLYCYCLOALKYL ALPHA-SUBSTITUTED TRP-PHE- AND PHENETHYLAMINE DERIVATIVES WARNER-LAMBERT COMPANY (US) 1991-01-10 WO disclosed
EP-0405537-A1 N-substituted cycloalkyl and polycycloalkyl alpha-substituted Trp-Phe- and phenethylamine derivatives WARNER-LAMBERT COMPANY (US) 1991-01-02 EP disclosed