SCHEMBL8716092

SCHEMBL8716092

COc1c(C(=O)N[C@H]2CC[C@H](OCC(=O)OC(C)(C)C)CC2)oc2ccc(C(=N)N)cc12

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.39
RAB9A P51151 3/20 0.39
F2 P00734 5/20 0.37
ITGB3 P05106 2/20 0.37
ITGA2B P08514 2/20 0.37
TPSAB1 Q15661 1/20 0.37
TPSD1 Q9BZJ3 1/20 0.37
TPSG1 Q9NRR2 1/20 0.37
HPGDS O60760 2/20 0.36
ST14 Q9Y5Y6 4/20 0.35
PRSS1 P07477 3/20 0.35
PRSS2 P07478 3/20 0.35
PRSS3 P35030 3/20 0.35
PLG P00747 1/20 0.35
CHRNB2 P17787 1/20 0.35
CHRNA7 P36544 1/20 0.35
CHRNA4 P43681 1/20 0.35
ALDH1A1 P00352 2/20 0.35
MEN1 O00255 1/20 0.35
HTT P42858 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8904086 1.00 NPC1 (0.39) NPC1RAB9AF2ITGB3ITGA2B
SCHEMBL8715011 0.90 NPC1 (0.46) NPC1RAB9AITGB3ITGA2BALDH1A1
SCHEMBL8906270 0.90 NPC1 (0.46) NPC1RAB9AITGB3ITGA2BALDH1A1
SCHEMBL8904560 0.89 ITGB3 (0.43) NPC1RAB9AF2ITGB3ITGA2B
SCHEMBL8713033 0.89 ITGB3 (0.43) NPC1RAB9AF2ITGB3ITGA2B
SCHEMBL8904093 0.86 ITGB3 (0.37) F2ITGB3ITGA2BTPSAB1TPSD1
SCHEMBL8904764 0.84 CETP (0.40) NPC1RAB9ACHRNB2CHRNA7CHRNA4
SCHEMBL8713211 0.84 CETP (0.40) NPC1RAB9ACHRNB2CHRNA7CHRNA4
SCHEMBL8906283 0.84 ITGB3 (0.40) F2ITGB3ITGA2BTPSAB1TPSD1
SCHEMBL8903361 0.82 F2 (0.51) NPC1RAB9AF2ITGB3ITGA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5753670-A ANTICOAGULANTS THE GREEN CROSS CORPORATION (JP) 1998-05-19 US disclosed
US-5635527-A ANTAGONIST OF PLATELET MEMBRANE GLYCOPROTEIN; TREATMENT OF THROMBOTIC DISEASES THE GREEN CROSS CORPORATION (JP) 1997-06-03 US disclosed
EP-0712844-A1 NOVEL FUSED-RING CARBOXYLIC ACID COMPOUND OR SALT THEREOF, AND MEDICINAL USE THEREOF THE GREEN CROSS CORPORATION (JP) 1996-05-22 EP disclosed