SCHEMBL8716754

SCHEMBL8716754

COc1cccc(CNC(=O)c2ccc(CO)cc2)c1

nearest known ligand 0.75

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MMP13 P45452 3/20 0.75
ROCK2 O75116 2/20 0.70
CYP3A4 P08684 1/20 0.70
CYP2D6 P10635 1/20 0.70
CYP2C9 P11712 1/20 0.70
PRKACA P17612 1/20 0.70
GSK3A P49840 1/20 0.70
GSK3B P49841 1/20 0.70
PRKX P51817 1/20 0.70
PRKCQ Q04759 1/20 0.70
ROCK1 Q13464 1/20 0.70
CLK4 Q9HAZ1 1/20 0.70
HPGD P15428 2/20 0.67
LMNA P02545 1/20 0.67
HDAC1 Q13547 1/20 0.64
MAPT P10636 1/20 0.62
ALDH1A1 P00352 3/20 0.61
GAA P10253 1/20 0.61
AURKA O14965 1/20 0.60
KDM4E B2RXH2 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8716430 0.88 MMP13 (0.73) MMP13ROCK2CYP3A4CYP2D6CYP2C9
SCHEMBL3816981 0.88 MMP13 (0.77) MMP13ROCK2CYP3A4CYP2D6CYP2C9
SCHEMBL13940425 0.88 MMP13 (0.90) MMP13ROCK2CYP3A4CYP2D6CYP2C9
SCHEMBL7134254 0.87 MMP13 (0.86) MMP13ROCK2CYP3A4CYP2D6CYP2C9
SCHEMBL31396722 0.86 MMP13 (0.75) MMP13ROCK2CYP3A4CYP2D6CYP2C9
SCHEMBL3816878 0.86 HPGD (0.79) MMP13ROCK2CYP3A4CYP2D6CYP2C9
SCHEMBL9416645 0.86 MMP13 (0.94) MMP13ROCK2CYP3A4CYP2D6CYP2C9
SCHEMBL31061610 0.86 MMP13 (1.00) MMP13ROCK2CYP3A4CYP2D6CYP2C9
SCHEMBL5332068 0.86 MMP13 (1.00) MMP13ROCK2CYP3A4CYP2D6CYP2C9
SCHEMBL17694837 0.85 EPHX2 (0.62) MMP13ROCK2ROCK1HPGDLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5728835-A HYPOTENSIVE AGENTS; ANTIISCHEMIC AGENTS TOA EIYO, LTD. (JP) 1998-03-17 US disclosed
EP-0661266-A1 Substituted cyclic amine compounds as 5HT2 antagonists TOA EIYO LTD. (JP) 1995-07-05 EP disclosed