SCHEMBL8716760

SCHEMBL8716760

COc1ccc(N(CCN2CCC(C(=O)c3ccc(F)cc3)CC2)C(=O)c2ccc(N(C)C(C)=O)cc2)cc1

nearest known ligand 0.54

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PTGIR P43119 1/20 0.54
OPRM1 P35372 1/20 0.53
ALDH1A1 P00352 1/20 0.52
LMNA P02545 1/20 0.52
HSD11B1 P28845 1/20 0.52
SMN1; SMN2 Q16637 1/20 0.52
SLC18A3 Q16572 6/20 0.48
DRD2 P14416 1/20 0.48
CYP1A2 P05177 1/20 0.48
GAA P10253 1/20 0.48
CYP2C9 P11712 1/20 0.48
CYP2C19 P33261 1/20 0.48
KMT2A Q03164 1/20 0.47
HTR2A P28223 1/20 0.47
HTR2C P28335 1/20 0.47
HTR7 P34969 1/20 0.47
HTR6 P50406 1/20 0.47
GLA P06280 1/20 0.46
MAPK1 P28482 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Fumaric Acid SCHEMBL8714261 0.95 PTGIR (0.51) PTGIROPRM1ALDH1A1LMNAHSD11B1
Fumaric Acid SCHEMBL8714256 0.95 PTGIR (0.51) PTGIROPRM1ALDH1A1LMNAHSD11B1
SCHEMBL8711220 0.92 PTGIR (0.56) PTGIROPRM1ALDH1A1LMNAHSD11B1
SCHEMBL8710939 0.91 HSD11B1 (0.52) PTGIROPRM1ALDH1A1LMNAHSD11B1
SCHEMBL8711336 0.89 PTGIR (0.55) PTGIROPRM1ALDH1A1LMNAHSD11B1
SCHEMBL8712161 0.88 CYP2C9 (0.58) PTGIROPRM1ALDH1A1LMNAHSD11B1
SCHEMBL8711249 0.88 PTGIR (0.54) PTGIROPRM1ALDH1A1LMNAHSD11B1
SCHEMBL8716637 0.88 PTGIR (0.54) PTGIROPRM1ALDH1A1LMNAHSD11B1
Fumaric Acid SCHEMBL8715314 0.87 PTGIR (0.54) PTGIROPRM1ALDH1A1LMNAHSD11B1
Fumaric Acid SCHEMBL8716585 0.86 HSD11B1 (0.47) PTGIROPRM1HSD11B1DRD2HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5728835-A HYPOTENSIVE AGENTS; ANTIISCHEMIC AGENTS TOA EIYO, LTD. (JP) 1998-03-17 US disclosed
EP-0661266-A1 Substituted cyclic amine compounds as 5HT2 antagonists TOA EIYO LTD. (JP) 1995-07-05 EP disclosed