SCHEMBL8718692

SCHEMBL8718692

CCOC(=O)Nc1c(C)c(C)c2c(c1C)CC(C)(C)O2

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 6/20 0.36
MEN1 O00255 2/20 0.36
HPGD P15428 2/20 0.36
NPSR1 Q6W5P4 1/20 0.36
EZH2 Q15910 1/20 0.35
KDM4E B2RXH2 2/20 0.35
GLA P06280 1/20 0.35
POLB P06746 1/20 0.35
NLRP3 Q96P20 3/20 0.35
CYP1A2 P05177 2/20 0.34
CYP2C9 P11712 2/20 0.34
CYP2C19 P33261 2/20 0.34
NPC1 O15118 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
HTT P42858 1/20 0.34
RAB9A P51151 1/20 0.34
ALDH1A1 P00352 3/20 0.34
LMNA P02545 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8718408 0.83 MEN1 (0.39) KMT2AMEN1HPGDEZH2KDM4E
SCHEMBL8875480 0.81 ALDH1A1 (0.41) KMT2AMEN1HPGDEZH2KDM4E
Hydrochloric Acid SCHEMBL8712939 0.80 ALDH1A1 (0.40) KMT2AMEN1HPGDEZH2KDM4E
Hydrochloric Acid SCHEMBL8717770 0.74 EZH2 (0.30) EZH2
SCHEMBL8720009 0.74 MAPT (0.44) KMT2AMEN1HPGDKDM4EPOLB
SCHEMBL8717999 0.72 MAPT (0.35) NPSR1KDM4EHTTALDH1A1LMNA
Hydrochloric Acid SCHEMBL8717929 0.70 HPGD (0.32) HPGD
SCHEMBL8714697 0.69 MEN1 (0.34) KMT2AMEN1EZH2POLBCYP1A2
SCHEMBL8713529 0.69 MEN1 (0.34) KMT2AMEN1HPGDEZH2KDM4E
SCHEMBL8718653 0.68 MEN1 (0.33) KMT2AMEN1EZH2POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5770772-A 4-FORMYLAMINO-2,3,5-TRIMETHYL-1-(2-METHYL-2-PROPENYLOXY) -BENZENE; ARTERIOSCLEROSIS, BRAIN AND CARDIOVASCULAR DISORDERS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-06-23 US disclosed
US-5594154-A 5-AMINO-2-BROMOMETHYL-2,4,6,7-TETRAMETHYL-2,3-DIHYDROBENZO(B) FURANS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-01-14 US disclosed
US-5478844-A Method of using aminocoumaran derivatives for treating cerebrovascular diseases TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1995-12-26 US disclosed
EP-0483772-B1 Aminocoumaran derivatives, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1995-09-13 EP disclosed
US-5376681-A Aminocoumaran derivatives, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1994-12-27 US disclosed
CN-1071165-A Aminocoumaran derivatives, their production and use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1993-04-21 CN disclosed
EP-0483772-A1 Aminocoumaran derivatives, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1992-05-06 EP disclosed