SCHEMBL8719347

SCHEMBL8719347

CC(C)(C)OC(=O)NCCCN(CCCCCCCN(CCCNC(=O)OC(C)(C)C)C(=O)OC(C)(C)C)C(=O)OC(C)(C)C

nearest known ligand 0.68

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CA14 Q9ULX7 1/20 0.68
TDP1 Q9NUW8 1/20 0.63
MEN1 O00255 1/20 0.51
GAA P10253 1/20 0.51
KMT2A Q03164 1/20 0.51
MAOA P21397 1/20 0.51
MAOB P27338 1/20 0.51
CA1 P00915 7/20 0.48
CA2 P00918 7/20 0.48
CA12 O43570 6/20 0.48
CA9 Q16790 6/20 0.48
STK17B O94768 1/20 0.41
STK17A Q9UEE5 1/20 0.41
EPHX1 P07099 1/20 0.39
HTT P42858 1/20 0.39
DRD2 P14416 1/20 0.39
CYP3A4 P08684 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8021860 1.00 CA14 (0.68) CA14TDP1MEN1GAAKMT2A
SCHEMBL13055412 0.97 CA14 (0.64) CA14TDP1MEN1GAAKMT2A
SCHEMBL13055410 0.97 CA14 (0.68) CA14TDP1MEN1GAAKMT2A
SCHEMBL8714161 0.97 CA14 (0.68) CA14TDP1MEN1GAAKMT2A
SCHEMBL31329717 0.94 TDP1 (0.69) CA14TDP1MEN1GAAKMT2A
SCHEMBL8020881 0.94 CA14 (0.60) CA14TDP1MEN1GAAKMT2A
SCHEMBL13055400 0.94 CA14 (0.64) CA14TDP1MEN1GAAKMT2A
SCHEMBL8850859 0.93 CA14 (0.60) CA14TDP1MEN1GAAKMT2A
SCHEMBL14439576 0.93 CA14 (0.60) CA14TDP1MEN1GAAKMT2A
SCHEMBL9885950 0.92 CA14 (0.63) CA14TDP1MEN1GAAKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0378146-A2 Polyamine derivatives as antineoplastic agents MERRELL PHARMACEUTICALS INC. (US) 1990-07-18 EP claimed
EP-0490380-B1 Use of N,N'-bis 3-(ethylamino)propyl -1,7-heptanediamine and a cytotoxic agent MERRELL PHARMA INC (US) 1998-02-18 EP disclosed
US-5654287-A SYNERGISTIC MERRELL PHAMACEUTICALS INC. (US) 1997-08-05 US disclosed
US-5646124-A ANTIBIOTIC MERRELL PHARMACEUTICALS INC. (US) 1997-07-08 US disclosed
US-5635218-A ADMINISTERING WITH ANTINEOPLASTIC PLATINUM COORDINATION COMPLEX; SYNERGISTIC EFFECT MERRELL PHARMACEUTICALS INC. (US) 1997-06-03 US disclosed
US-5561136-A USING VINBLASTINE AS SYNERGISTIC CYTOTOXIC AGENT MERRELL PHARMACEUTICALS INC. (US) 1996-10-01 US disclosed
EP-0662829-A1 POLYAMINE DERIVATIVES AS ANTI-CYTOMEGALOVIRAL AGENTS MERRELL PHARMACEUTICALS INC. (US) 1995-07-19 EP disclosed
EP-0378146-B1 Polyamine derivatives as antineoplastic agents MERRELL DOW PHARMA (US) 1995-03-29 EP disclosed
WO-1994007480-A1 POLYAMINE DERIVATIVES AS ANTI-CYTOMEGALOVIRAL AGENTS MERRELL DOW PHARMACEUTICALS INC. (US) 1994-04-14 WO disclosed
EP-0490380-A2 Use of N,N'-bis 3-(ethylamino)propyl -1,7-heptanediamine and a cytotoxic agent MERRELL PHARMACEUTICALS INC. (US) 1992-06-17 EP disclosed
US-5109024-A Polyamine derivatives as antineoplastic agents MERRELL DOW PHARMACEUTICALS INC. (US) 1992-04-28 US disclosed
EP-0378146-A2 Polyamine derivatives as antineoplastic agents MERRELL PHARMACEUTICALS INC. (US) 1990-07-18 EP disclosed