SCHEMBL8719970

SCHEMBL8719970

O=C(NC[C@@H]1CCCNC1)c1ccccc1

nearest known ligand 0.60

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.60
CHEK1 O14757 2/20 0.55
NAMPT P43490 1/20 0.55
PBK Q96KB5 5/20 0.54
SMN1; SMN2 Q16637 1/20 0.54
HPGD P15428 1/20 0.51
CTSL P07711 1/20 0.50
CTSB P07858 1/20 0.50
CTSK P43235 1/20 0.50
ACP1 P24666 1/20 0.50
SMYD3 Q9H7B4 2/20 0.49
MEN1 O00255 1/20 0.49
CHRM2 P08172 1/20 0.48
CHRM3 P20309 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2423748 1.00 KMT2A (0.60) KMT2ACHEK1NAMPTPBKSMN1; SMN2
SCHEMBL8719751 1.00 KMT2A (0.60) KMT2ACHEK1NAMPTPBKSMN1; SMN2
SCHEMBL5094284 0.91 NAMPT (0.63) KMT2ANAMPTSMN1; SMN2HPGDCTSL
SCHEMBL13325381 0.91 NAMPT (0.63) KMT2ANAMPTSMN1; SMN2HPGDCTSL
SCHEMBL13325386 0.91 NAMPT (0.63) KMT2ANAMPTSMN1; SMN2HPGDCTSL
Mandelic Acid SCHEMBL8716945 0.89 KMT2A (0.50) KMT2ACHEK1NAMPTPBKSMN1; SMN2
Mandelic Acid SCHEMBL7303904 0.89 KMT2A (0.50) KMT2ACHEK1NAMPTPBKSMN1; SMN2
Mandelic Acid SCHEMBL7297870 0.89 KMT2A (0.50) KMT2ACHEK1NAMPTPBKSMN1; SMN2
Mandelic Acid SCHEMBL7303720 0.89 KMT2A (0.50) KMT2ACHEK1NAMPTPBKSMN1; SMN2
Mandelic Acid SCHEMBL8716949 0.89 KMT2A (0.50) KMT2ACHEK1NAMPTPBKSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-109476633-A The inhibitor of tryptophan 2,3- dioxygenase 荷兰转化研究中心有限责任公司 2019-03-15 CN disclosed
US-5763604-A ANTICOAGULANTS HOFFMANN-LA ROCHE INC. (US) 1998-06-09 US disclosed
US-5677448-A CHEMICAL INTERMEDIATES FOR MAKING ANTAGONIST OF THROMBIN, TREATING THROMBOSIS, STROKE, INFLAMMATION, ARTERIOSCLEROSIS, CARDIOVASCULAR DISORDERS HOFFMANN-LA ROCHE INC. (US) 1997-10-14 US disclosed
US-5578594-A ANTICOAGULANTS HOFFMANN-LA ROCHE INC. (US) 1996-11-26 US disclosed
US-5405854-A Anticoagulants HOFFMANN-LA ROCHE INC. (US) 1995-04-11 US disclosed
CN-1076690-A SULFONAMIDOCARBOXAMIDES HOFFMANN LA ROCHE (CH) 1993-09-29 CN disclosed