SCHEMBL5094284

SCHEMBL5094284

O=C(NCC1CCNC1)c1ccccc1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 3/20 0.63
SMYD3 Q9H7B4 3/20 0.57
CTSL P07711 1/20 0.52
CTSB P07858 1/20 0.52
CTSK P43235 1/20 0.52
HPGD P15428 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
ITGB3 P05106 1/20 0.49
ITGA2B P08514 1/20 0.49
OPRM1 P35372 1/20 0.49
KDM1A O60341 1/20 0.49
MAOB P27338 1/20 0.49
KMT2A Q03164 1/20 0.49
KDM4E B2RXH2 1/20 0.48
PKM P14618 1/20 0.48
HDAC3 O15379 1/20 0.48
HDAC4 P56524 1/20 0.48
HDAC1 Q13547 1/20 0.48
HDAC7 Q8WUI4 1/20 0.48
HDAC2 Q92769 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13325381 1.00 NAMPT (0.63) NAMPTSMYD3CTSLCTSBCTSK
SCHEMBL13325386 1.00 NAMPT (0.63) NAMPTSMYD3CTSLCTSBCTSK
SCHEMBL2423748 0.91 KMT2A (0.60) NAMPTSMYD3CTSLCTSBCTSK
SCHEMBL8719970 0.91 KMT2A (0.60) NAMPTSMYD3CTSLCTSBCTSK
SCHEMBL8719751 0.91 KMT2A (0.60) NAMPTSMYD3CTSLCTSBCTSK
SCHEMBL3330915 0.91 SMN1; SMN2 (0.56) NAMPTSMYD3CTSLCTSBCTSK
SCHEMBL4956356 0.89 CTSL (0.59) NAMPTCTSLCTSBCTSKHPGD
SCHEMBL17888454 0.85 SMYD3 (0.58) NAMPTSMYD3OPRM1KDM1AKMT2A
SCHEMBL8255991 0.85 SMYD3 (0.58) NAMPTSMYD3OPRM1
SCHEMBL14720114 0.85 SMYD3 (0.58) NAMPTSMYD3HPGDKMT2AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-2008516973-A 2008-05-22 JP claimed
EP-1812439-A2 KINASE INHIBITORS Takeda San Diego, Inc. (US) 2007-08-01 EP claimed
WO-2006044687-A2 KINASE INHIBITORS TAKEDA SAN DIEGO, INC. (US) 2006-04-27 WO claimed
EP-1765789-B1 N-(1-(1-BENZYL-4-PHENYL-1H-IMIDAZOL-2-YL)-2,2-DIMETHYLPROPYL)BENZAMIDE DERIVATIVES AND RELATED COMPOUNDS AS KINESIN SPINDLE PROTEIN (KSP) INHIBITORS FOR THE TREATMENT OF CANCER NOVARTIS AG (CH) 2013-02-27 EP disclosed
EP-1812439-A2 KINASE INHIBITORS Takeda San Diego, Inc. (US) 2007-08-01 EP disclosed
WO-2006044687-A2 KINASE INHIBITORS TAKEDA SAN DIEGO, INC. (US) 2006-04-27 WO disclosed