SCHEMBL8720641

SCHEMBL8720641

COc1c(Cl)cc(O)cc1Cl

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.56
CYP3A4 P08684 4/20 0.54
MAPT P10636 1/20 0.54
HPGD P15428 3/20 0.50
HSD17B10 Q99714 3/20 0.50
CRHBP P24387 1/20 0.50
CRHR2 Q13324 1/20 0.50
ALDH1A1 P00352 4/20 0.48
KDM4E B2RXH2 2/20 0.48
GAA P10253 2/20 0.48
TPMT P51580 1/20 0.48
TAS1R3 Q7RTX0 3/20 0.41
TAS1R1 Q7RTX1 3/20 0.41
TAS1R2 Q8TE23 3/20 0.41
KMT2A Q03164 2/20 0.40
MEN1 O00255 1/20 0.40
LMNA P02545 1/20 0.40
HTT P42858 1/20 0.40
CHRM1 P11229 1/20 0.40
ALOX15 P16050 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2388019 0.86 CYP3A4 (0.71) TDP1CYP3A4MAPTHPGDHSD17B10
SCHEMBL12745843 0.84 TDP1 (0.46) TDP1CYP3A4MAPTHPGDHSD17B10
SCHEMBL4119971 0.80 ALDH1A1 (0.49) TDP1CYP3A4MAPTHPGDHSD17B10
SCHEMBL28610832 0.80 ERN1 (0.46) TDP1CYP3A4MAPTALDH1A1KDM4E
SCHEMBL9331998 0.79 TPMT (0.48) TDP1CYP3A4MAPTHPGDHSD17B10
SCHEMBL24516637 0.78 GALK1 (0.50) TDP1MAPTHPGDHSD17B10ALDH1A1
SCHEMBL9617366 0.78 CYP3A4 (0.48) TDP1CYP3A4MAPTHPGDHSD17B10
SCHEMBL54507 0.78 KMT2A (0.47) TDP1CYP3A4MAPTHPGDHSD17B10
SCHEMBL12325399 0.78 ALDH1A1 (0.47) TDP1HPGDHSD17B10ALDH1A1KDM4E
SCHEMBL9623900 0.78 HSD17B10 (0.55) TDP1CYP3A4MAPTHPGDHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0662004-B1 USE OF PERSISTENT FREE-RADICALS IN MAGNETIC RESONANCE IMAGING NYCOMED INNOVATION AB (SE) 1998-03-18 EP disclosed
US-5700448-A Use of persistent free-radicals in magnetic resonance imaging NYCOMED IMAGING AS (NO) 1997-12-23 US disclosed
US-5435991-A Use of persistent heterocyclic free-radicals in magnetic resonance imaging NYCOMED INNOVATION AB (SE) 1995-07-25 US disclosed
EP-0662004-A1 USE OF PERSISTENT FREE-RADICALS IN MAGNETIC RESONANCE IMAGING Nycomed Innovation AB (SE) 1995-07-12 EP disclosed
WO-1993002710-A2 USE OF PERSISTENT FREE RADICALS IN MAGNETIC RESONANCE IMAGING NYCOMED INNOVATION AB (SE) 1993-02-18 WO disclosed
WO-1993002711-A1 USE OF PERSISTENT FREE-RADICALS IN MAGNETIC RESONANCE IMAGING NYCOMED INNOVATION AB (SE) 1993-02-18 WO disclosed