SCHEMBL8723377

SCHEMBL8723377

Cc1[nH]nc(C(=N)N)c1C

nearest known ligand 0.42

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
DYRK1A Q13627 1/20 0.42
HCAR2 Q8TDS4 3/20 0.36
KIT P10721 3/20 0.31
AKT2 P31751 1/20 0.31
KMT2A Q03164 1/20 0.31
HTT P42858 1/20 0.30
PTK2 Q05397 1/20 0.30
CSNK2A2 P19784 1/20 0.30
KDR P35968 1/20 0.30
CSNK2B P67870 1/20 0.30
CSNK2A1 P68400 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL599727 0.77 HCAR2 (0.45) DYRK1AHCAR2KITCSNK2A2KDR
SCHEMBL9123806 0.74 HCAR2 (0.39) HCAR2CSNK2A2KDRCSNK2BCSNK2A1
SCHEMBL4631308 0.70 HCAR2 (0.63) DYRK1AHCAR2
SCHEMBL6195861 0.68 PDE4D (0.47) DYRK1AAKT2CSNK2A2KDRCSNK2B
SCHEMBL600381 0.67
Hydrochloric Acid SCHEMBL15550505 0.65
SCHEMBL20798457 0.65 HCAR2 (0.42) DYRK1AHCAR2KIT
SCHEMBL459546 0.64 DYRK1A (0.42) DYRK1A
SCHEMBL19158730 0.63 PDE4D (0.59) HCAR2KITKMT2A
SCHEMBL14190551 0.62 HCAR2 (0.44) HCAR2CSNK2A2KDRCSNK2BCSNK2A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0879227-A1 TYROSIN-DERIVATE AS ALPHA-V-INTEGRIN INHIBITORS MERCK PATENT GmbH (DE) 1998-11-25 EP disclosed
WO-1997023451-A1 TYROSIN-DERIVATE AS ALPHA-V-INTEGRIN INHIBITORS MERCK Patent Gesellschaft mit beschränkter Haftung (DE) 1997-07-03 WO disclosed