SCHEMBL8724358

SCHEMBL8724358

Cc1cc(C)cc(C(=O)N[C@H](Cc2ccccc2)C(=O)N[C@@H](Cc2c[nH]c3ccccc23)C(=O)O)c1

nearest known ligand 0.70

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 4/20 0.70
ITGB2 P05107 2/20 0.66
ICAM1 P05362 2/20 0.66
ITGAL P20701 2/20 0.66
PLAU P00749 1/20 0.63
PLAUR Q03405 1/20 0.63
ERAP2 Q6P179 1/20 0.62
ACE P12821 2/20 0.60
LTA4H P09960 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8724361 1.00 TACR1 (0.70) TACR1ITGB2ICAM1ITGALPLAU
SCHEMBL16617905 0.90 CTSL (0.67) TACR1ITGB2ICAM1ITGALPLAU
SCHEMBL16617908 0.90 CTSL (0.67) TACR1ITGB2ICAM1ITGALPLAU
SCHEMBL21427023 0.90 ITGB2 (0.70) TACR1ITGB2ICAM1ITGALPLAU
SCHEMBL23118282 0.89 TACR1 (0.59) TACR1ITGB2ICAM1ITGALPLAU
SCHEMBL23118287 0.89 EDNRB (0.60) TACR1ITGB2ICAM1ITGALPLAU
SCHEMBL29197301 0.89 ITGB2 (0.66) ITGB2ICAM1ITGALPLAUPLAUR
SCHEMBL8721736 0.87 EDNRB (0.77) TACR1ITGB2ICAM1ITGALPLAU
SCHEMBL23118288 0.87 EDNRB (0.58) TACR1ITGB2ICAM1ITGALPLAU
SCHEMBL11227413 0.85 CTSL (0.61) TACR1ITGB2ICAM1ITGALPLAU

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5780498-A PEPTIDE DERIVATIVES FOR CARDIOVASCULAR AND BRAIN DISORDERS CIBA-GEIGY JAPAN LIMITED (JP) 1998-07-14 US disclosed
WO-1995012611-A1 ENDOTHELIN RECEPTOR ANTAGONISTS JAPAT LTD. (CH) 1995-05-11 WO disclosed