SCHEMBL8724906

SCHEMBL8724906

C=Cc1c[c]c2c(C=C)cccc2c1

nearest known ligand 0.35

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.35
TP53 P04637 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
ALDH1A1 P00352 3/20 0.31
TSHR P16473 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7793839 0.73 ALDH1A1 (0.35) ALDH1A1
SCHEMBL7790730 0.72 ALDH1A1 (0.39) PARP1TP53TDP1ALDH1A1TSHR
SCHEMBL12986970 0.68 TP53 (0.41) PARP1TP53TDP1ALDH1A1TSHR
SCHEMBL29592963 0.68 TP53 (0.41) PARP1TP53TDP1ALDH1A1TSHR
SCHEMBL3850055 0.65 ALDH1A1 (0.32) ALDH1A1
SCHEMBL2443320 0.64 TYMS (0.42) TP53TDP1ALDH1A1TSHR
SCHEMBL16289143 0.64 ALDH1A1 (0.34) ALDH1A1
SCHEMBL29760312 0.64 TYMS (0.42) TP53TDP1ALDH1A1TSHR
SCHEMBL3807899 0.63 PPARG (0.44) TDP1ALDH1A1TSHR
SCHEMBL278142 0.62 ALDH1A1 (0.45) PARP1TP53TDP1ALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0609058-B1 Hexahydronaphthalene ester derivatives, their preparation and their therapeutic uses SANKYO CO (JP) 1998-12-09 EP disclosed
US-5491167-A INHIBITORS OF CHOLESTEROL BIOSYNTHESIS SANKYO COMPANY, LIMITED (JP) 1996-02-13 US disclosed
EP-0609058-A2 Hexahydronaphthalene ester derivatives, their preparation and their therapeutic uses SANKYO COMPANY LIMITED (JP) 1994-08-03 EP disclosed