SCHEMBL8725864

SCHEMBL8725864

CCOc1ccc(Nc2cc[c]cc2)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NQO1 P15559 1/20 0.54
GAA P10253 1/20 0.53
KDM4E B2RXH2 3/20 0.51
NFKB1 P19838 1/20 0.51
MAPT P10636 5/20 0.50
CTDSP1 Q9GZU7 1/20 0.50
ALDH1A1 P00352 3/20 0.49
LMNA P02545 2/20 0.49
TDP1 Q9NUW8 2/20 0.49
L3MBTL1 Q9Y468 2/20 0.49
NSD2 O96028 1/20 0.49
HPGD P15428 1/20 0.49
MAPK1 P28482 1/20 0.49
HTT P42858 1/20 0.49
SYK P43405 2/20 0.49
KMT2A Q03164 4/20 0.49
POLB P06746 3/20 0.49
MEN1 O00255 2/20 0.49
CYP1A2 P05177 1/20 0.49
OPRM1 P35372 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL49554 0.88 NQO1 (0.70) NQO1GAAKDM4ENFKB1MAPT
SCHEMBL9514574 0.88 NQO1 (0.70) NQO1GAAKDM4ENFKB1MAPT
SCHEMBL8721610 0.85 MAPT (0.50) GAAKDM4EMAPTALDH1A1TDP1
SCHEMBL21151 0.81
SCHEMBL8721616 0.80 KDM4E (0.44) GAAKDM4EMAPTTDP1L3MBTL1
SCHEMBL9479637 0.80 MAPT (0.63) NQO1GAAKDM4ENFKB1MAPT
SCHEMBL3627657 0.80 MAPT (0.71) NQO1GAAKDM4ENFKB1MAPT
SCHEMBL8738419 0.80 NQO1 (0.58) NQO1KDM4ENFKB1MAPTCTDSP1
SCHEMBL3440767 0.80 MAPT (0.63) NQO1GAAKDM4ENFKB1MAPT
SCHEMBL11677967 0.79 GAA (0.56) NQO1GAAKDM4ENFKB1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0832091-A1 C-4' MODIFIED ADENOSINE KINASE INHIBITORS GENSIA, INC. (US) 1998-04-01 EP disclosed
WO-1996040705-A1 C-4' MODIFIED ADENOSINE KINASE INHIBITORS GENSIA SICOR (US) 1996-12-19 WO disclosed