SCHEMBL8727581

SCHEMBL8727581

O=C(O)C(I)(CI)c1ccc(O)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 6/20 0.42
ESR2 Q92731 6/20 0.42
CYP3A4 P08684 4/20 0.42
ALDH1A1 P00352 2/20 0.42
CPT1B Q92523 1/20 0.39
BLM P54132 2/20 0.38
CA2 P00918 2/20 0.38
CES2 O00748 1/20 0.38
CAMK2A Q9UQM7 1/20 0.38
TYR P14679 2/20 0.37
LMNA P02545 1/20 0.37
AR P10275 1/20 0.37
HPGD P15428 1/20 0.37
TSHR P16473 1/20 0.37
SLC6A2 P23975 1/20 0.37
SLC6A4 P31645 1/20 0.37
HTR6 P50406 1/20 0.37
ESRRG P62508 1/20 0.37
SLC6A3 Q01959 1/20 0.37
HSD17B10 Q99714 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10458795 0.72 ESR1 (0.44) ESR1ESR2CYP3A4ALDH1A1BLM
SCHEMBL9644070 0.71 ESR1 (0.50) ESR1ESR2CYP3A4ALDH1A1CPT1B
SCHEMBL8727572 0.69 ESR1 (0.47) ESR1ESR2CYP3A4ALDH1A1BLM
SCHEMBL8028384 0.69 ESR1 (0.48) ESR1ESR2CYP3A4ALDH1A1BLM
SCHEMBL4206889 0.69 CA2 (0.48) ESR1ESR2CYP3A4ALDH1A1CPT1B
SCHEMBL31647379 0.68 BLM (0.42) ESR1ESR2CYP3A4ALDH1A1CPT1B
SCHEMBL4220470 0.67 ESR1 (0.44) ESR1ESR2CYP3A4ALDH1A1CPT1B
SCHEMBL9153305 0.67 ESR1 (0.44) ESR1ESR2CYP3A4ALDH1A1CPT1B
SCHEMBL24288076 0.66 ESR1 (0.54) ESR1ESR2CYP3A4ALDH1A1TYR
SCHEMBL9792726 0.66 CYP1A2 (0.43) ESR1ESR2CYP3A4ALDH1A1CPT1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0831769-A2 NOVEL USES FOR THYROID HORMONES OR THYROID HORMONE-LIKE COMPOUNDS KARO BIO AB (SE) 1998-04-01 EP claimed
WO-1996040048-A9 NOVEL USES FOR THYROID HORMONES OR THYROID HORMONE-LIKE COMPOUNDS 1997-03-27 WO claimed
WO-1996040048-A2 NOVEL USES FOR THYROID HORMONES OR THYROID HORMONE-LIKE COMPOUNDS KARO BIO AB (SE) 1996-12-19 WO claimed