SCHEMBL8728729

SCHEMBL8728729

COc1ccc(CCN(C)C)cc1OCc1ccccc1

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.72
CYP1A2 P05177 2/20 0.72
CYP3A4 P08684 2/20 0.72
CYP2D6 P10635 2/20 0.72
BLM P54132 2/20 0.72
CYP2C9 P11712 1/20 0.72
KMT2A Q03164 3/20 0.66
MEN1 O00255 2/20 0.66
SIGMAR1 Q99720 2/20 0.57
EBP Q15125 1/20 0.57
TMEM97 Q5BJF2 1/20 0.57
ABCB1 P08183 2/20 0.56
ABCG2 Q9UNQ0 1/20 0.56
LMNA P02545 2/20 0.55
HTT P42858 2/20 0.55
SMN1; SMN2 Q16637 2/20 0.55
NPY1R P25929 1/20 0.55
NPY2R P49146 1/20 0.55
BCHE P06276 1/20 0.55
PMP22 Q01453 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8734889 0.99 KDM4E (0.70) KDM4ECYP1A2CYP3A4CYP2D6BLM
SCHEMBL19194551 0.84 KDM4E (0.59) KDM4ECYP1A2CYP3A4CYP2D6BLM
SCHEMBL20079681 0.84 KDM4E (0.61) KDM4ECYP1A2CYP3A4CYP2D6BLM
SCHEMBL10118317 0.83 CYP1A2 (0.79) KDM4ECYP1A2CYP3A4CYP2D6BLM
SCHEMBL12296058 0.82 BCHE (0.61) KDM4ECYP1A2CYP3A4CYP2D6BLM
SCHEMBL2742565 0.82 KDM4E (0.68) KDM4ECYP1A2CYP3A4CYP2D6BLM
Hydrochloric Acid SCHEMBL17821823 0.81 KDM4E (0.66) KDM4ECYP1A2CYP3A4CYP2D6BLM
SCHEMBL8554822 0.80 MAPK1 (0.64) KDM4ECYP1A2CYP3A4CYP2D6BLM
SCHEMBL30472718 0.80 ABCB1 (0.59) KDM4ECYP1A2CYP3A4CYP2D6BLM
SCHEMBL9416643 0.80 KDM4E (0.81) KDM4ECYP1A2CYP3A4CYP2D6BLM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0641766-B1 ALKOXYPHENYLALKYLAMINE DERIVATIVE TAISHO PHARMACEUTICAL CO LTD (JP) 1998-11-11 EP disclosed
US-5495046-A PSYCHOLOGICAL DISORDERS TAISHO PHARMACEUTICAL CO., LTD. (JP) 1996-02-27 US disclosed
EP-0641766-A1 ALKOXYPHENYLALKYLAMINE DERIVATIVE TAISHO PHARMACEUTICAL CO. LTD (JP) 1995-03-08 EP disclosed