SCHEMBL9416643

SCHEMBL9416643

COc1cc(CN(C)Cc2ccc(OC)c(OCc3ccccc3)c2)ccc1OCc1ccccc1

nearest known ligand 0.81

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.81
CYP1A2 P05177 1/20 0.81
CYP3A4 P08684 1/20 0.81
CYP2D6 P10635 1/20 0.81
CYP2C9 P11712 1/20 0.81
BLM P54132 1/20 0.81
KMT2A Q03164 3/20 0.78
MEN1 O00255 2/20 0.78
NPC1 O15118 1/20 0.57
RAB9A P51151 1/20 0.57
MAPK1 P28482 1/20 0.57
HSD17B10 Q99714 1/20 0.57
BCHE P06276 4/20 0.56
ACHE P22303 2/20 0.56
ABCB1 P08183 2/20 0.56
ABCG2 Q9UNQ0 1/20 0.56
GAA P10253 1/20 0.55
MAPT P10636 1/20 0.55
APP P05067 2/20 0.54
LMNA P02545 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8782844 0.87 KDM4E (0.73) KDM4ECYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL28312736 0.86 KDM4E (0.64) KDM4ECYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL9416658 0.83 MEN1 (0.61) KDM4ECYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL2060386 0.82 MAPK1 (0.63) KDM4ECYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL3232932 0.82 MEN1 (0.64) KDM4ECYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL31388315 0.82 MEN1 (0.64) KDM4ECYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL9416623 0.81 HTT (0.61) KDM4ECYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL9416662 0.81 HTT (0.61) KDM4ECYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL9416614 0.81 LMNA (0.73) KDM4EKMT2AMEN1NPC1RAB9A
Bromide SCHEMBL20482559 0.81 MAPK1 (0.61) KDM4ECYP1A2CYP3A4CYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0613879-A1 PHELLODENDRINE ANALOGS AND ALLERGY TYPE IV SUPPRESSOR CONTAINING THE SAME AS ACTIVE INGREDIENT TSUMURA & CO. (JP) 1994-09-07 EP disclosed